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Found 57 Enz. Inhib. hit(s) with all data for entry = 50042439
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50098577(Benzofuran-2-carboxylic acid {3-methyl-1-[3-oxo-1-...)
Affinity DataKi:  0.160nMAssay Description:Inhibition of human cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50408519(CHEMBL115357)
Affinity DataKi:  0.700nMAssay Description:Inhibition of human cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM12042((2R,3R)-3-{[(1S)-1-[(4-carbamimidamidobutyl)carbam...)
Affinity DataKi:  1.40nMAssay Description:Inhibition of human cathepsin K by gelatin zymographic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM19807(CHEMBL100563 | benzyl N-[(1S)-1-({1-[(2S)-2-{[(ben...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of cathepsin K (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426169(CHEMBL2316589)
Affinity DataKi:  3.5nMAssay Description:Inhibition of cathepsin K (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50066648(((S)-3-Methyl-1-{3-[(S)-4-methyl-2-(pyridin-4-ylme...)
Affinity DataKi:  3.5nMAssay Description:Inhibition of cathepsin K (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50079596(((S)-1-{N'-[2-((S)-1-Benzyloxycarbonylamino-3-meth...)
Affinity DataKi:  10nMAssay Description:Inhibition of human cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426167(CHEMBL2316590)
Affinity DataKi:  12nMAssay Description:Inhibition of human cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426170(CHEMBL2316313)
Affinity DataKi:  13nMAssay Description:Inhibition of cathepsin K (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50066650(1,3-BIS[[N-[(PHENYLMETHOXY)CARBONYL]-L-LEUCYL]AMIN...)
Affinity DataKi:  22nMAssay Description:Inhibition of cathepsin K (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426168(CHEMBL2316303)
Affinity DataIC50:  0.25nMAssay Description:Inhibition of cathepsin K (unknown origin)More data for this Ligand-Target Pair
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426166(CHEMBL2316304)
Affinity DataIC50:  0.830nMAssay Description:Inhibition of human cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50137816(((S)-1-Cyclohexyl-2-oxo-ethyl)-carbamic acid tert-...)
Affinity DataIC50:  26nMAssay Description:Inhibition of cathepsin K (unknown origin)More data for this Ligand-Target Pair
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426157(CHEMBL2316613)
Affinity DataIC50:  100nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50303426(4-(isopropylamino)-6-(phenylamino)-1,3,5-triazine-...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426153(CHEMBL1355124)
Affinity DataIC50:  400nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426127(CHEMBL2316307)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426132(CHEMBL2316606)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426138(CHEMBL2316600)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426139(CHEMBL1620957)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426159(CHEMBL2311590)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426146(CHEMBL1419509)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426150(CHEMBL2316593)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426130(CHEMBL2316305)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426143(CHEMBL2316598)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426136(2-(1-Cyclododecylethylidene)Hydrazinecarbothioamid...)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426128(CHEMBL2316306)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426135(CHEMBL2316603)
Affinity DataIC50:  1.05E+4nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426133(CHEMBL2316605)
Affinity DataIC50:  1.33E+4nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426125(CHEMBL2316309)
Affinity DataIC50:  1.81E+4nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426161(CHEMBL2316610)
Affinity DataIC50:  1.93E+4nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426164(CHEMBL2316608)
Affinity DataIC50:  1.96E+4nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426158(CHEMBL2316612)
Affinity DataIC50:  2.13E+4nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426123(CHEMBL2316311)
Affinity DataIC50:  2.14E+4nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426165(CHEMBL1432431)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426163(CHEMBL1319029)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426162(CHEMBL2316609)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426160(CHEMBL2316611)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426156(CHEMBL2316614)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426155(2-(3-(Phenylsulfonyl)Allylthio)Benzo[D]Thiazole | ...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426154(CHEMBL2316616)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426152(CHEMBL1526900)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426151(CHEMBL2316592)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426149(CHEMBL2316594)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426148(CHEMBL2316595)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426147(CHEMBL1863593)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426145(CHEMBL2316596)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426144(CHEMBL2316597)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426142(CHEMBL1341853)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Msd Animal Health Innovation

Curated by ChEMBL
LigandPNGBDBM50426141(CHEMBL2316599)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant His-tagged cathepsin K using Cbz-Phe-Arg-AMC as substrate incubated for 30 mins prior to substrate addition by FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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