Compile Data Set for Download or QSAR
maximum 50k data
Found 127 Enz. Inhib. hit(s) with all data for entry = 50042712
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429823(CHEMBL2338173)
Affinity DataKi:  0.150nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429823(CHEMBL2338173)
Affinity DataKi:  6.80nMAssay Description:Binding affinity to CB1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429830(CHEMBL2338182)
Affinity DataKi:  170nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429829(CHEMBL2338183)
Affinity DataKi:  200nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429826(CHEMBL2338186)
Affinity DataKi:  270nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429824(CHEMBL2338188)
Affinity DataKi:  320nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429835(CHEMBL2338176)
Affinity DataKi:  350nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429826(CHEMBL2338186)
Affinity DataKi:  400nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429833(CHEMBL2338178)
Affinity DataKi:  460nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429832(CHEMBL2338179)
Affinity DataKi:  500nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429834(CHEMBL2338177)
Affinity DataKi:  500nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429825(CHEMBL2338187)
Affinity DataKi:  500nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429831(CHEMBL2338181)
Affinity DataKi:  500nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429827(CHEMBL2338185)
Affinity DataKi:  600nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429837(CHEMBL2338174)
Affinity DataKi:  770nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50207795(CHEMBL246952 | adamantan-1-yl-(3,4-dihydro-2H-quin...)
Affinity DataKi:  790nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429832(CHEMBL2338179)
Affinity DataKi:  900nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429836(CHEMBL2338175)
Affinity DataKi:  990nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429830(CHEMBL2338182)
Affinity DataKi:  1.30E+3nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429835(CHEMBL2338176)
Affinity DataKi:  1.50E+3nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429824(CHEMBL2338188)
Affinity DataKi:  2.20E+3nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429829(CHEMBL2338183)
Affinity DataKi:  2.40E+3nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429828(CHEMBL2338184)
Affinity DataKi:  2.50E+3nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429828(CHEMBL2338184)
Affinity DataKi:  2.80E+3nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429834(CHEMBL2338177)
Affinity DataKi:  2.80E+3nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50207795(CHEMBL246952 | adamantan-1-yl-(3,4-dihydro-2H-quin...)
Affinity DataKi:  4.30E+3nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429831(CHEMBL2338181)
Affinity DataKi:  4.90E+3nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429837(CHEMBL2338174)
Affinity DataKi:  5.20E+3nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429836(CHEMBL2338175)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429833(CHEMBL2338178)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429827(CHEMBL2338185)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429825(CHEMBL2338187)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Mus musculus (Mouse))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429824(CHEMBL2338188)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Mus musculus (Mouse))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429825(CHEMBL2338187)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Mus musculus (Mouse))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429826(CHEMBL2338186)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Mus musculus (Mouse))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429827(CHEMBL2338185)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Mus musculus (Mouse))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429828(CHEMBL2338184)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Mus musculus (Mouse))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429829(CHEMBL2338183)
Affinity DataEC50: >6.00E+3nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Mus musculus (Mouse))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429830(CHEMBL2338182)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Mus musculus (Mouse))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429831(CHEMBL2338181)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Mus musculus (Mouse))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429832(CHEMBL2338179)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Mus musculus (Mouse))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429833(CHEMBL2338178)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Mus musculus (Mouse))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429834(CHEMBL2338177)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Mus musculus (Mouse))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429835(CHEMBL2338176)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Mus musculus (Mouse))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429836(CHEMBL2338175)
Affinity DataEC50:  5.00E+3nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429834(CHEMBL2338177)
Affinity DataEC50:  22nMAssay Description:Agonist activity at mouse CB2 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429835(CHEMBL2338176)
Affinity DataEC50:  20nMAssay Description:Agonist activity at mouse CB2 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429837(CHEMBL2338174)
Affinity DataEC50:  23nMAssay Description:Agonist activity at mouse CB2 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50207795(CHEMBL246952 | adamantan-1-yl-(3,4-dihydro-2H-quin...)
Affinity DataEC50:  126nMAssay Description:Agonist activity at mouse CB2 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50429838(CHEMBL2338189)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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