Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with all data for entry = 50042548
TargetGlutamate receptor 2(Homo sapiens (Human))
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50427677(CHEMBL2323527)
Affinity DataKi:  5.60E+5nMAssay Description:Binding affinity to GluA2 ligand binding domain (unknown origin) by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
Yokohama City University

Curated by ChEMBL
LigandPNGBDBM50178141((S)-1-(2-amino-2-carboxyethyl)-3-(4-carboxybenzyl)...)
Affinity DataIC50:  2.90E+5nMAssay Description:Displacement of [3H]AMPA from rat GluA2 ligand binding domain after 1 hrMore data for this Ligand-Target Pair