Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50005423
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Central South University

Curated by ChEMBL
LigandPNGBDBM50491979(CHEMBL2392467)
Affinity DataIC50:  470nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin) assessed as inhibition of MEK phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Central South University

Curated by ChEMBL
LigandPNGBDBM50491978(CHEMBL2392604)
Affinity DataIC50:  630nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin) assessed as inhibition of MEK phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Central South University

Curated by ChEMBL
LigandPNGBDBM50491976(CHEMBL2392599)
Affinity DataIC50:  770nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin) assessed as inhibition of MEK phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Central South University

Curated by ChEMBL
LigandPNGBDBM50491975(CHEMBL2392473)
Affinity DataIC50:  1.16E+3nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin) assessed as inhibition of MEK phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Central South University

Curated by ChEMBL
LigandPNGBDBM50491977(CHEMBL2392468)
Affinity DataIC50:  2.01E+3nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin) assessed as inhibition of MEK phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Central South University

Curated by ChEMBL
LigandPNGBDBM50491980(CHEMBL2392569)
Affinity DataIC50:  2.16E+3nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin) assessed as inhibition of MEK phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed