Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 50042901
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50432942(CHEMBL2377721)
Affinity DataIC50:  33nMAssay Description:Inhibition of human full length Pim-3 using RSRHSSYPAGT as substrate assessed as residual activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50432946(CHEMBL2377711)
Affinity DataIC50:  119nMAssay Description:Inhibition of human full length Pim-3 using RSRHSSYPAGT as substrate assessed as residual activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50432946(CHEMBL2377711)
Affinity DataIC50:  230nMAssay Description:Inhibition of human full length Pim-1 using RSRHSSYPAGT as substrate assessed as residual activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50432945(CHEMBL2377716)
Affinity DataIC50:  260nMAssay Description:Inhibition of human full length Pim-3 using RSRHSSYPAGT as substrate assessed as residual activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50432942(CHEMBL2377721)
Affinity DataIC50:  460nMAssay Description:Inhibition of human full length Pim-1 using RSRHSSYPAGT as substrate assessed as residual activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50432947(CHEMBL2377724)
Affinity DataIC50:  470nMAssay Description:Inhibition of human full length Pim-3 using RSRHSSYPAGT as substrate assessed as residual activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50432943(CHEMBL2377718)
Affinity DataIC50:  530nMAssay Description:Inhibition of human full length Pim-3 using RSRHSSYPAGT as substrate assessed as residual activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50432944(CHEMBL2377717)
Affinity DataIC50:  546nMAssay Description:Inhibition of human full length Pim-3 using RSRHSSYPAGT as substrate assessed as residual activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50432943(CHEMBL2377718)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human full length Pim-1 using RSRHSSYPAGT as substrate assessed as residual activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed