Compile Data Set for Download or QSAR
maximum 50k data
Found 46 Enz. Inhib. hit(s) with all data for entry = 50044052
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004891(CHEMBL2164327)
Affinity DataKi:  0.600nMAssay Description:Binding affinity to human 5HT7 receptor expressed in HEK-293F cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50098551((R)-3-(2-(2-(4-methylpiperidin-1-yl)ethyl)pyrrolid...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to 5HT7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50001888((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50001888((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50098550(3,N-Dimethyl-N-[(R)-1-methyl-3-(4-methyl-piperidin...)
Affinity DataKi:  32nMAssay Description:Binding affinity to 5HT7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004894(CHEMBL2376461)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004894(CHEMBL2376461)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004892(CHEMBL2375370)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004892(CHEMBL2375370)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004893(CHEMBL2376462)
Affinity DataKi:  77nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004893(CHEMBL2376462)
Affinity DataKi:  77nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004898(CHEMBL2376458)
Affinity DataKi:  219nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004898(CHEMBL2376458)
Affinity DataKi:  219nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004896(CHEMBL2376459)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004896(CHEMBL2376459)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004900(CHEMBL2376457)
Affinity DataKi:  297nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004900(CHEMBL2376457)
Affinity DataKi:  297nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004895(CHEMBL2376460)
Affinity DataKi:  311nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004895(CHEMBL2376460)
Affinity DataKi:  311nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004909(CHEMBL2376469)
Affinity DataKi:  432nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004909(CHEMBL2376469)
Affinity DataKi:  432nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004890(CHEMBL2376463)
Affinity DataKi:  537nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004890(CHEMBL2376463)
Affinity DataKi:  537nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004902(CHEMBL2376456)
Affinity DataKi:  658nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004902(CHEMBL2376456)
Affinity DataKi:  658nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004905(CHEMBL2376449)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004905(CHEMBL2376449)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004903(CHEMBL2376455)
Affinity DataKi:  1.66E+3nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004903(CHEMBL2376455)
Affinity DataKi:  1.66E+3nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004906(CHEMBL2376448)
Affinity DataKi:  1.75E+3nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004906(CHEMBL2376448)
Affinity DataKi:  1.75E+3nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004908(CHEMBL2376447)
Affinity DataKi:  1.85E+3nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004908(CHEMBL2376447)
Affinity DataKi:  1.85E+3nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004904(CHEMBL2376450)
Affinity DataKi:  2.76E+3nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004904(CHEMBL2376450)
Affinity DataKi:  2.76E+3nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004928(CHEMBL2376466)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004911(CHEMBL2376453)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004910(CHEMBL2376454)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004889(CHEMBL2376464)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004914(CHEMBL2376471)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004912(CHEMBL2376452)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004929(CHEMBL2376465)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004916(CHEMBL2376468)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004926(CHEMBL2376467)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004913(CHEMBL2376451)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50004915(CHEMBL2376470)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-LSD from 5HT7 receptor (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed