Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with all data for entry = 50005277
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mahidol University

Curated by ChEMBL
LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of HIV-1 reverse transcriptase assessed as decrease in incorporation of [3H]TTP into polyA templateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50478514(Fagaronine | Fagaronine Chloride)
Affinity DataIC50:  2.65E+4nMAssay Description:Inhibition of HIV-1 reverse transcriptase assessed as decrease in incorporation of [3H]TTP into polyA templateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50490558(Dikamaliartane D)
Affinity DataIC50:  6.87E+4nMAssay Description:Inhibition of HIV-1 reverse transcriptase assessed as decrease in incorporation of [3H]TTP into polyA templateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50490559(CHEMBL2332127 | Rel-Carinatin C)
Affinity DataIC50:  8.57E+4nMAssay Description:Inhibition of HIV-1 reverse transcriptase assessed as decrease in incorporation of [3H]TTP into polyA templateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed