Compile Data Set for Download or QSAR
maximum 50k data
Found 15 Enz. Inhib. hit(s) with all data for entry = 7303
TargetPantothenate kinase(Mycobacterium tuberculosis ATCC 25618/H37Rv)
Uppsala University

LigandPNGBDBM188493(Triazole 1e)
Affinity DataIC50:  50nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
TargetPantothenate kinase(Mycobacterium tuberculosis ATCC 25618/H37Rv)
Uppsala University

LigandPNGBDBM188489(Triazole 1a)
Affinity DataIC50:  90nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
TargetPantothenate kinase(Mycobacterium tuberculosis ATCC 25618/H37Rv)
Uppsala University

LigandPNGBDBM188495(Biaryl 2a)
Affinity DataIC50:  120nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPantothenate kinase(Mycobacterium tuberculosis ATCC 25618/H37Rv)
Uppsala University

LigandPNGBDBM188495(Biaryl 2a)
Affinity DataIC50:  130nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPantothenate kinase(Mycobacterium tuberculosis ATCC 25618/H37Rv)
Uppsala University

LigandPNGBDBM188492(Triazole 1d)
Affinity DataIC50:  140nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
TargetPantothenate kinase(Mycobacterium tuberculosis ATCC 25618/H37Rv)
Uppsala University

LigandPNGBDBM188491(Triazole 1c)
Affinity DataIC50:  150nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPantothenate kinase(Mycobacterium tuberculosis ATCC 25618/H37Rv)
Uppsala University

LigandPNGBDBM188496(Biaryl 2b)
Affinity DataIC50:  550nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPantothenate kinase(Mycobacterium tuberculosis ATCC 25618/H37Rv)
Uppsala University

LigandPNGBDBM188493(Triazole 1e)
Affinity DataIC50:  690nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
TargetPantothenate kinase(Mycobacterium tuberculosis ATCC 25618/H37Rv)
Uppsala University

LigandPNGBDBM188494(Triazole 1f)
Affinity DataIC50:  1.09E+3nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
TargetPantothenate kinase(Mycobacterium tuberculosis ATCC 25618/H37Rv)
Uppsala University

LigandPNGBDBM188490(Triazole 1b)
Affinity DataIC50:  1.13E+3nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
TargetPantothenate kinase(Mycobacterium tuberculosis ATCC 25618/H37Rv)
Uppsala University

LigandPNGBDBM188492(Triazole 1d)
Affinity DataIC50:  2.82E+3nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
TargetPantothenate kinase(Mycobacterium tuberculosis ATCC 25618/H37Rv)
Uppsala University

LigandPNGBDBM188489(Triazole 1a)
Affinity DataIC50:  5.50E+3nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
TargetPantothenate kinase(Mycobacterium tuberculosis ATCC 25618/H37Rv)
Uppsala University

LigandPNGBDBM188491(Triazole 1c)
Affinity DataIC50:  1.04E+4nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPantothenate kinase(Mycobacterium tuberculosis ATCC 25618/H37Rv)
Uppsala University

LigandPNGBDBM188490(Triazole 1b)
Affinity DataIC50: >1.25E+4nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair
TargetPantothenate kinase(Mycobacterium tuberculosis ATCC 25618/H37Rv)
Uppsala University

LigandPNGBDBM188494(Triazole 1f)
Affinity DataIC50:  1.40E+4nMAssay Description:Briefly, MtPanK activity was measured in a pyruvate kinaselactate dehydrogenase-coupled assay where the reaction rate was determined by spectrophotom...More data for this Ligand-Target Pair