Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50043350
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM81395(APO-866)
Affinity DataKi:  0.300nMAssay Description:Noncompetitive inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50439676(CHEMBL2417796)
Affinity DataIC50:  0.230nMAssay Description:Inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50347432(CHEMBL1801863)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50347433(CHEMBL1801864)
Affinity DataIC50:  0.450nMAssay Description:Inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50439675(CHEMBL2417788 | US11279687, Compound 196)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50439678(CHEMBL2417789)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of recombinant his-tagged NAMPT (unknown origin) expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50439677(CHEMBL2417790 | US9169209, Table 3, Compound 55)
Affinity DataIC50:  3nMAssay Description:Inhibition of recombinant his-tagged NAMPT (unknown origin) expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50439680(CHEMBL2417798)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of recombinant his-tagged NAMPT (unknown origin) expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50439679(CHEMBL2417799)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of recombinant his-tagged NAMPT (unknown origin) expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50005031(CHEMBL2417792)
Affinity DataIC50: <5.00E+3nMAssay Description:Inhibition of NAMPT in human U87 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50439681(CHEMBL2417797)
Affinity DataKd:  4.50E+4nMAssay Description:Binding affinity to NAMPT (unknown origin)More data for this Ligand-Target Pair