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Found 29 Enz. Inhib. hit(s) with all data for entry = 50043221
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50369323(MECAMYLAMINE)
Affinity DataIC50:  600nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437522(CHEMBL2407120)
Affinity DataIC50:  6.00E+3nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437521(CHEMBL2407121)
Affinity DataIC50:  7.50E+3nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50366799(TUBOCURARINE | TUBOCURARINE CHLORIDE)
Affinity DataIC50:  9.20E+3nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437513(CHEMBL2407128)
Affinity DataIC50:  1.48E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437534(CHEMBL2407134)
Affinity DataIC50:  1.54E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437518(CHEMBL152025)
Affinity DataIC50:  1.71E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437517(CHEMBL2407124)
Affinity DataIC50:  1.93E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437519(CHEMBL2407123)
Affinity DataIC50:  1.94E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437520(CHEMBL2407122)
Affinity DataIC50:  1.96E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437514(CHEMBL2407127)
Affinity DataIC50:  2.05E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437512(CHEMBL2407129)
Affinity DataIC50:  2.24E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437536(CHEMBL2407132)
Affinity DataIC50:  2.32E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437535(CHEMBL2407133)
Affinity DataIC50:  3.76E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437533(CHEMBL2407135)
Affinity DataIC50:  5.41E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437516(CHEMBL2407125)
Affinity DataIC50:  7.01E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437511(CHEMBL2407130)
Affinity DataIC50:  8.07E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437526(CHEMBL2409791)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437527(CHEMBL2407141)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437528(CHEMBL2407140)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437529(CHEMBL2407139)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437530(CHEMBL2407138)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437531(CHEMBL2407137)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437532(CHEMBL2407136)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437510(CHEMBL2407131)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437525(CHEMBL2409792)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437524(CHEMBL2409793)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437515(CHEMBL2407126)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437523(CHEMBL2409794)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed