TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Competitive inhibition of Pin1 (unknown origin) by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Reversible inhibition of human Pin1More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of GST-tagged Pin1 (unknown origin) using Suc-AEPF-pNA and WFYpSPR-pNA as substrate after 5 minsMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of human Pin1More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 890nMAssay Description:Inhibition of human Pin1More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Reversible inhibition of human Pin1More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of Pin1 (unknown origin) using Suc-Ala-Glu-cis-Pro-Phe-pNA as substrateMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of Pin1 (unknown origin) using Suc-Ala-Glu-Pro-Phe-MCA as substrate after 120 secs by fluorescence microtiter plate reader analysisMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 4(Homo sapiens (Human))
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of Par14 (unknown origin)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of human Pin1More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 6.10E+3nMAssay Description:Binding affinity to GST-tagged Pin1 (unknown origin) by SPR spectroscopic analysisMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human Pin1More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of full length Pin1 (unknown origin) using WFY(pS)PR-pNA as substrate by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataKd: 1.50E+4nMAssay Description:Binding affinity to Pin1 WW domain (unknown origin)More data for this Ligand-Target Pair