Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50043276
TargetD(2) dopamine receptor(Homo sapiens (Human))
Columbia University Medical Center

Curated by ChEMBL
LigandPNGBDBM50438565(CHEMBL2413153)
Affinity DataKi:  37nMAssay Description:Binding affinity to dopamine 2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Columbia University Medical Center

Curated by ChEMBL
LigandPNGBDBM86757(CAS_0 | NSC_11603174 | [11C]MMP)
Affinity DataKi:  59nMAssay Description:Binding affinity to sigma 1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Columbia University Medical Center

Curated by ChEMBL
LigandPNGBDBM50438565(CHEMBL2413153)
Affinity DataKi:  512nMAssay Description:Binding affinity to histamine H1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Columbia University Medical Center

Curated by ChEMBL
LigandPNGBDBM86757(CAS_0 | NSC_11603174 | [11C]MMP)
Affinity DataKi:  1.03E+3nMAssay Description:Binding affinity to histamine H1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
Columbia University Medical Center

Curated by ChEMBL
LigandPNGBDBM50438565(CHEMBL2413153)
Affinity DataKi:  1.77E+3nMAssay Description:Binding affinity to histamine H2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
Columbia University Medical Center

Curated by ChEMBL
LigandPNGBDBM86757(CAS_0 | NSC_11603174 | [11C]MMP)
Affinity DataKi:  2.13E+3nMAssay Description:Binding affinity to histamine H2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Columbia University Medical Center

Curated by ChEMBL
LigandPNGBDBM50438565(CHEMBL2413153)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to sigma 1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Columbia University Medical Center

Curated by ChEMBL
LigandPNGBDBM86757(CAS_0 | NSC_11603174 | [11C]MMP)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to dopamine 2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed