Compile Data Set for Download or QSAR
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Found 32 Enz. Inhib. hit(s) with all data for entry = 50043277
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438573(CHEMBL2413705)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438573(CHEMBL2413705)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438581(CHEMBL448807)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438576(CHEMBL2413704)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438581(CHEMBL448807)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438567(CHEMBL512713)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438568(CHEMBL2413710)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438576(CHEMBL2413704)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438575(CHEMBL486977)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438574(CHEMBL486969)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438566(CHEMBL2413711)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438568(CHEMBL2413710)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438571(CHEMBL2413707)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438580(CHEMBL2413700)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438575(CHEMBL486977)
Affinity DataIC50:  1.05E+5nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438571(CHEMBL2413707)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438566(CHEMBL2413711)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438569(CHEMBL2413709)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438570(CHEMBL2413708)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438572(CHEMBL2413706)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438570(CHEMBL2413708)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438574(CHEMBL486969)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438569(CHEMBL2413709)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438577(CHEMBL2413703)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438578(CHEMBL2413702)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438579(CHEMBL2413701)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438567(CHEMBL512713)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438577(CHEMBL2413703)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438580(CHEMBL2413700)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438572(CHEMBL2413706)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438578(CHEMBL2413702)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Aston University

Curated by ChEMBL
LigandPNGBDBM50438579(CHEMBL2413701)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed