Found 89 Enz. Inhib. hit(s) with all data for entry = 50043252 
Affinity DataIC50: 6nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataIC50: 6nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 41nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 76nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 89nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 147nMAssay Description:Inhibition of human PARP1 catalytic activity after 10 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataKd: 1.00E+4nMAssay Description:Binding affinity to catalytic domain of human PARP1 after 5 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
Affinity DataKd: 46nMAssay Description:Binding affinity to catalytic domain of human PARP1 after 5 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
Affinity DataKd: 296nMAssay Description:Binding affinity to catalytic domain of human PARP1 after 5 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
Affinity DataKd: 96nMAssay Description:Binding affinity to catalytic domain of human PARP1 after 5 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.50E+4nMAssay Description:Binding affinity to catalytic domain of human PARP1 after 5 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
Affinity DataKd: 5.20E+3nMAssay Description:Binding affinity to catalytic domain of human PARP1 after 5 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+4nMAssay Description:Binding affinity to catalytic domain of human PARP1 after 5 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
Affinity DataKd: 2.60E+4nMAssay Description:Binding affinity to catalytic domain of human PARP1 after 5 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.00E+5nMAssay Description:Binding affinity to catalytic domain of human PARP1 after 5 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.70E+5nMAssay Description:Binding affinity to catalytic domain of human PARP1 after 5 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
Affinity DataKd: >5.00E+5nMAssay Description:Binding affinity to catalytic domain of human PARP1 after 5 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
Affinity DataKd: 3.20E+4nMAssay Description:Binding affinity to catalytic domain of human PARP1 after 5 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
Affinity DataKd: >5.00E+5nMAssay Description:Binding affinity to catalytic domain of human PARP1 after 5 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Inhibition of PARP1 in human Jurkat cells assessed as reduction of cell viability after 96 hrs by MTS assay in presence of 100 uM of temozolomideMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+4nMAssay Description:Inhibition of PARP1 in human Jurkat cells assessed as reduction of cell viability after 96 hrs by MTS assay in presence of 100 uM of temozolomideMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+4nMAssay Description:Inhibition of PARP1 in human Jurkat cells assessed as reduction of cell viability after 96 hrs by MTS assay in presence of 100 uM of temozolomideMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60E+4nMAssay Description:Inhibition of PARP1 in human Jurkat cells assessed as reduction of cell viability after 96 hrs by MTS assay in presence of 100 uM of temozolomideMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60E+4nMAssay Description:Inhibition of PARP1 in human Jurkat cells assessed as reduction of cell viability after 96 hrs by MTS assay in presence of 100 uM of temozolomideMore data for this Ligand-Target Pair
Affinity DataEC50: 2.70E+4nMAssay Description:Inhibition of PARP1 in human Jurkat cells assessed as reduction of cell viability after 96 hrs by MTS assay in presence of 100 uM of temozolomideMore data for this Ligand-Target Pair
Affinity DataEC50: 5.00E+3nMAssay Description:Inhibition of PARP1 in human Jurkat cells assessed as reduction of cell viability after 96 hrs by MTS assay in presence of 100 uM of temozolomideMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+5nMAssay Description:Inhibition of PARP1 in human Jurkat cells assessed as reduction of cell viability after 96 hrs by MTS assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.60E+4nMAssay Description:Inhibition of PARP1 in human Jurkat cells assessed as reduction of cell viability after 96 hrs by MTS assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7.70E+4nMAssay Description:Inhibition of PARP1 in human Jurkat cells assessed as reduction of cell viability after 96 hrs by MTS assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.40E+4nMAssay Description:Inhibition of PARP1 in human Jurkat cells assessed as reduction of cell viability after 96 hrs by MTS assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+5nMAssay Description:Inhibition of PARP1 in human Jurkat cells assessed as reduction of cell viability after 96 hrs by MTS assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+5nMAssay Description:Inhibition of PARP1 in human Jurkat cells assessed as reduction of cell viability after 96 hrs by MTS assayMore data for this Ligand-Target Pair
