Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 6010
TargetSerine/threonine-protein kinase PKH2 [1-944](Candida albicans SC5314)
Universit£Tsklinikum Frankfurt

LigandPNGBDBM104016(PS77)
Affinity DataIC50:  1.70E+4nMpH: 7.4 T: 2°CAssay Description:A 20ul mix containing 50mM Tris pH 7.5, 0.05mg/ml BSA, 0.1% β-mercaptoethanol, 10mM MgCl2, 100μM [γ-P32]ATP (5-50cpm/pmol), 0.003% Bri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Universit£Tsklinikum Frankfurt

LigandPNGBDBM104018(PS182)
Affinity DataIC50:  2.60E+4nMpH: 7.4 T: 2°CAssay Description:The AlphaScreen Assay (Perkin Elmer) was performed according to the manufacturer's protocol in 384-well microtiter plates. Incubations were performe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Universit£Tsklinikum Frankfurt

LigandPNGBDBM104016(PS77)
Affinity DataIC50:  3.80E+4nMpH: 7.4 T: 2°CAssay Description:A 20ul mix containing 50mM Tris pH 7.5, 0.05mg/ml BSA, 0.1% β-mercaptoethanol, 10mM MgCl2, 100μM [γ-P32]ATP (5-50cpm/pmol), 0.003% Bri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Universit£Tsklinikum Frankfurt

LigandPNGBDBM50399646(CHEMBL2177668 | PS210)
Affinity DataIC50:  3.90E+4nMpH: 7.4 T: 2°CAssay Description:The AlphaScreen Assay (Perkin Elmer) was performed according to the manufacturer's protocol in 384-well microtiter plates. Incubations were performe...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Universit£Tsklinikum Frankfurt

LigandPNGBDBM50296949((2Z)-5-(4-chlorophenyl)-3-phenylpent-2-enoic acid ...)
Affinity DataIC50:  9.70E+4nMpH: 7.4 T: 2°CAssay Description:The AlphaScreen Assay (Perkin Elmer) was performed according to the manufacturer's protocol in 384-well microtiter plates. Incubations were performe...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PKH2 [1-944](Candida albicans SC5314)
Universit£Tsklinikum Frankfurt

LigandPNGBDBM104018(PS182)
Affinity DataEC50:  6.60E+4nMpH: 7.4 T: 2°CAssay Description:The AlphaScreen Assay (Perkin Elmer) was performed according to the manufacturer's protocol in 384-well microtiter plates. Incubations were performe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PKH2 [1-944](Candida albicans SC5314)
Universit£Tsklinikum Frankfurt

LigandPNGBDBM50321382(2-(3-(4-chlorophenyl)-3-oxo-1-phenylpropylthio)ace...)
Affinity DataEC50:  8.50E+4nMpH: 7.4 T: 2°CAssay Description:The AlphaScreen Assay (Perkin Elmer) was performed according to the manufacturer's protocol in 384-well microtiter plates. Incubations were performe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PKH2 [1-944](Candida albicans SC5314)
Universit£Tsklinikum Frankfurt

LigandPNGBDBM104016(PS77)
Affinity DataEC50:  4.40E+4nMpH: 7.4Assay Description:The AlphaScreen Assay (Perkin Elmer) was performed according to the manufacturer's protocol in 384-well microtiter plates. Incubations were performe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PKH2 [1-944](Candida albicans SC5314)
Universit£Tsklinikum Frankfurt

LigandPNGBDBM50399646(CHEMBL2177668 | PS210)
Affinity DataEC50:  6.00E+4nMpH: 7.4 T: 2°CAssay Description:The AlphaScreen Assay (Perkin Elmer) was performed according to the manufacturer's protocol in 384-well microtiter plates. Incubations were performe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed