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Found 22 Enz. Inhib. hit(s) with all data for entry = 50043324
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50439350(CHEMBL2420385)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human recombinant IRAP expressed in HeLa cells assessed as L-Leucine-7-amido-4-methyl coumarin hydrolysis to 7-amido-4-methyl coumarin ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50439354(CHEMBL2420381)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of recombinant ERAP1 (unknown origin) expressed in baculovirus-infected Hi5 insect cells assessed as L-Leucine-7-amido-4-methyl coumarin h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50439353(CHEMBL2420382)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of recombinant ERAP1 (unknown origin) expressed in baculovirus-infected Hi5 insect cells assessed as L-Leucine-7-amido-4-methyl coumarin h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50439351(CHEMBL2420384)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of human recombinant IRAP expressed in HeLa cells assessed as L-Leucine-7-amido-4-methyl coumarin hydrolysis to 7-amido-4-methyl coumarin ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50439357(CHEMBL2420378)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of human recombinant IRAP expressed in HeLa cells assessed as L-Leucine-7-amido-4-methyl coumarin hydrolysis to 7-amido-4-methyl coumarin ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50439353(CHEMBL2420382)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of human recombinant IRAP expressed in HeLa cells assessed as L-Leucine-7-amido-4-methyl coumarin hydrolysis to 7-amido-4-methyl coumarin ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50439351(CHEMBL2420384)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of recombinant ERAP1 (unknown origin) expressed in baculovirus-infected Hi5 insect cells assessed as L-Leucine-7-amido-4-methyl coumarin h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50439353(CHEMBL2420382)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus-infected Hi5 insect cells assessed as L-Arginyl-7-amido-4-methyl coumarin h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50439352(CHEMBL2420383)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of human recombinant IRAP expressed in HeLa cells assessed as L-Leucine-7-amido-4-methyl coumarin hydrolysis to 7-amido-4-methyl coumarin ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50439354(CHEMBL2420381)
Affinity DataIC50:  1.03E+4nMAssay Description:Inhibition of human recombinant IRAP expressed in HeLa cells assessed as L-Leucine-7-amido-4-methyl coumarin hydrolysis to 7-amido-4-methyl coumarin ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50439357(CHEMBL2420378)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus-infected Hi5 insect cells assessed as L-Arginyl-7-amido-4-methyl coumarin h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50439349(CHEMBL2420386)
Affinity DataIC50:  1.63E+4nMAssay Description:Inhibition of human recombinant IRAP expressed in HeLa cells assessed as L-Leucine-7-amido-4-methyl coumarin hydrolysis to 7-amido-4-methyl coumarin ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50439350(CHEMBL2420385)
Affinity DataIC50:  2.39E+4nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus-infected Hi5 insect cells assessed as L-Arginyl-7-amido-4-methyl coumarin h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50439354(CHEMBL2420381)
Affinity DataIC50:  2.49E+4nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus-infected Hi5 insect cells assessed as L-Arginyl-7-amido-4-methyl coumarin h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50439358(CHEMBL2420377)
Affinity DataIC50:  3.83E+4nMAssay Description:Inhibition of human recombinant IRAP expressed in HeLa cells assessed as L-Leucine-7-amido-4-methyl coumarin hydrolysis to 7-amido-4-methyl coumarin ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50439355(CHEMBL2420380)
Affinity DataIC50:  4.60E+4nMAssay Description:Inhibition of human recombinant IRAP expressed in HeLa cells assessed as L-Leucine-7-amido-4-methyl coumarin hydrolysis to 7-amido-4-methyl coumarin ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50439357(CHEMBL2420378)
Affinity DataIC50:  9.55E+4nMAssay Description:Inhibition of recombinant ERAP1 (unknown origin) expressed in baculovirus-infected Hi5 insect cells assessed as L-Leucine-7-amido-4-methyl coumarin h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50439351(CHEMBL2420384)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus-infected Hi5 insect cells assessed as L-Arginyl-7-amido-4-methyl coumarin h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50439348(CHEMBL2420387)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus-infected Hi5 insect cells assessed as L-Arginyl-7-amido-4-methyl coumarin h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50439356(CHEMBL2420379)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant IRAP expressed in HeLa cells assessed as L-Leucine-7-amido-4-methyl coumarin hydrolysis to 7-amido-4-methyl coumarin ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50439348(CHEMBL2420387)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant IRAP expressed in HeLa cells assessed as L-Leucine-7-amido-4-methyl coumarin hydrolysis to 7-amido-4-methyl coumarin ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50439349(CHEMBL2420386)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus-infected Hi5 insect cells assessed as L-Arginyl-7-amido-4-methyl coumarin h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed