Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50043476
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Capital Normal University

Curated by ChEMBL
LigandPNGBDBM50441661(CHEMBL2435034)
Affinity DataIC50:  240nMAssay Description:Inhibition of TGFbeta-induced downstream transcriptional activation of ALK5 (unknown origin) expressed in CHO-HIR cells assessed as intracellular tra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Capital Normal University

Curated by ChEMBL
LigandPNGBDBM50110208(4-(4-(benzo[d][1,3]dioxol-5-yl)-5-(pyridin-2-yl)-1...)
Affinity DataIC50:  350nMAssay Description:Inhibition of TGFbeta-induced downstream transcriptional activation of ALK5 (unknown origin) expressed in CHO-HIR cells assessed as intracellular tra...More data for this Ligand-Target Pair
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Capital Normal University

Curated by ChEMBL
LigandPNGBDBM50441660(CHEMBL2435035)
Affinity DataIC50:  650nMAssay Description:Inhibition of TGFbeta-induced downstream transcriptional activation of ALK5 (unknown origin) expressed in CHO-HIR cells assessed as intracellular tra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Capital Normal University

Curated by ChEMBL
LigandPNGBDBM50441659(CHEMBL2435036)
Affinity DataIC50:  800nMAssay Description:Inhibition of TGFbeta-induced downstream transcriptional activation of ALK5 (unknown origin) expressed in CHO-HIR cells assessed as intracellular tra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Capital Normal University

Curated by ChEMBL
LigandPNGBDBM50441662(CHEMBL2435041)
Affinity DataIC50:  950nMAssay Description:Inhibition of TGFbeta-induced downstream transcriptional activation of ALK5 (unknown origin) expressed in CHO-HIR cells assessed as intracellular tra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Capital Normal University

Curated by ChEMBL
LigandPNGBDBM50441666(CHEMBL2435044)
Affinity DataIC50:  990nMAssay Description:Inhibition of TGFbeta-induced downstream transcriptional activation of ALK5 (unknown origin) expressed in CHO-HIR cells assessed as intracellular tra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Capital Normal University

Curated by ChEMBL
LigandPNGBDBM50441663(CHEMBL2435040)
Affinity DataIC50:  1.78E+3nMAssay Description:Inhibition of TGFbeta-induced downstream transcriptional activation of ALK5 (unknown origin) expressed in CHO-HIR cells assessed as intracellular tra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Capital Normal University

Curated by ChEMBL
LigandPNGBDBM50441664(CHEMBL2435039)
Affinity DataIC50:  2.08E+3nMAssay Description:Inhibition of TGFbeta-induced downstream transcriptional activation of ALK5 (unknown origin) expressed in CHO-HIR cells assessed as intracellular tra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Capital Normal University

Curated by ChEMBL
LigandPNGBDBM50441667(CHEMBL2435043)
Affinity DataIC50:  2.43E+3nMAssay Description:Inhibition of TGFbeta-induced downstream transcriptional activation of ALK5 (unknown origin) expressed in CHO-HIR cells assessed as intracellular tra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Capital Normal University

Curated by ChEMBL
LigandPNGBDBM50441665(CHEMBL2435045)
Affinity DataIC50:  3.36E+3nMAssay Description:Inhibition of TGFbeta-induced downstream transcriptional activation of ALK5 (unknown origin) expressed in CHO-HIR cells assessed as intracellular tra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Capital Normal University

Curated by ChEMBL
LigandPNGBDBM50441658(CHEMBL2435037)
Affinity DataIC50:  3.82E+3nMAssay Description:Inhibition of TGFbeta-induced downstream transcriptional activation of ALK5 (unknown origin) expressed in CHO-HIR cells assessed as intracellular tra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed