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Found 21 Enz. Inhib. hit(s) with all data for entry = 50043573
TargetCytochrome P450 2D6(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50443210(CHEMBL3087352)
Affinity DataIC50:  100nMAssay Description:Inhibition of CYP2D6 (unknown origin) after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50443208(CHEMBL3087355)
Affinity DataIC50:  200nMAssay Description:Inhibition of CYP2D6 (unknown origin) after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50443202(CHEMBL3087041)
Affinity DataIC50:  700nMAssay Description:Inhibition of CYP2D6 (unknown origin) after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50443201(CHEMBL3087042)
Affinity DataIC50:  700nMAssay Description:Inhibition of CYP2D6 (unknown origin) after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50443200(CHEMBL3087043)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of CYP2D6 (unknown origin) after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50443203(CHEMBL3087040)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of CYP2D6 (unknown origin) after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50443204(CHEMBL3087038)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of CYP2D6 (unknown origin) after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50443195(CHEMBL3087343)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of CYP2D6 (unknown origin) after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50443215(CHEMBL3087347)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of CYP2D6 (unknown origin) after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50443196(CHEMBL3087342)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of CYP2D6 (unknown origin) after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50443206(CHEMBL3087036)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of CYP2D6 (unknown origin) after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50443205(CHEMBL3087037)
Affinity DataIC50:  9.80E+3nMAssay Description:Inhibition of CYP2D6 (unknown origin) after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50443211(CHEMBL3087351)
Affinity DataIC50:  1.18E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin) after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50443197(CHEMBL3087341)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin) after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50443213(CHEMBL3087349)
Affinity DataIC50:  1.51E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin) after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50443212(CHEMBL3087350)
Affinity DataIC50: >2.70E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin) after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50443207(CHEMBL3087035)
Affinity DataIC50: >2.70E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin) after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50443214(CHEMBL3087348)
Affinity DataIC50: >2.70E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin) after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50443198(CHEMBL3087340)
Affinity DataIC50: >2.70E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin) after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50443209(CHEMBL3087353)
Affinity DataIC50: >2.70E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin) after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50443199(CHEMBL3087339)
Affinity DataIC50: >2.70E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin) after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed