Compile Data Set for Download or QSAR
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Found 9 Enz. Inhib. hit(s) with all data for entry = 50043593
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443388(CHEMBL3086782 | US9688668, SLR080811)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of sphingosine kinase 1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443385(SPC-100270 | Safingol | Safingol HCl)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of sphingosine kinase 1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443389(CHEMBL2376441)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of sphingosine kinase 1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443384(CHEMBL3086799)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of recombinant sphingosine kinase 1 (unknown origin) expressed in HEK293 cells using sphingosine as substrate after 30 mins in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443387(CHEMBL3086811)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of recombinant sphingosine kinase 1 (unknown origin) expressed in HEK293 cells using sphingosine as substrate after 30 mins in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443383(CHEMBL3086796)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of sphingosine kinase 2 (unknown origin) using sphingosine as substrate after 30 mins in presence of [gamma32P]-ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443384(CHEMBL3086799)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of sphingosine kinase 2 (unknown origin) using sphingosine as substrate after 30 mins in presence of [gamma32P]-ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443383(CHEMBL3086796)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of recombinant sphingosine kinase 1 (unknown origin) expressed in HEK293 cells using sphingosine as substrate after 30 mins in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443386(CHEMBL3086806)
Affinity DataIC50:  1.69E+4nMAssay Description:Inhibition of recombinant sphingosine kinase 1 (unknown origin) expressed in HEK293 cells using sphingosine as substrate after 30 mins in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed