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Found 67 Enz. Inhib. hit(s) with all data for entry = 50005781
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494431(CHEMBL3087715)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494430(CHEMBL3087716)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494427(CHEMBL3087707)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494425(CHEMBL3087706)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494425(CHEMBL3087706)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494431(CHEMBL3087715)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494423(CHEMBL3087717)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494429(CHEMBL3087711)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50256890(8-Bromo-9-ethyl-9H-adenine | CHEMBL468633)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494433(CHEMBL3087713)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494424(CHEMBL3087710)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494427(CHEMBL3087707)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494430(CHEMBL3087716)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494423(CHEMBL3087717)
Affinity DataKi:  69nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50257054(8-Bromo-9-(3-hydroxypropyl)-9H-adenine | CHEMBL475...)
Affinity DataKi:  85nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494428(CHEMBL3087712)
Affinity DataKi:  89nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494426(CHEMBL3087714)
Affinity DataKi:  106nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494434(CHEMBL3087708)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50256842(8-Bromo-9-methyl-9H-adenine | CHEMBL510288)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494424(CHEMBL3087710)
Affinity DataKi:  193nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50256893(8-Bromo-9-propyl-9H-adenine | CHEMBL506450)
Affinity DataKi:  200nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494425(CHEMBL3087706)
Affinity DataKi:  250nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50256890(8-Bromo-9-ethyl-9H-adenine | CHEMBL468633)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50256893(8-Bromo-9-propyl-9H-adenine | CHEMBL506450)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494427(CHEMBL3087707)
Affinity DataKi:  350nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494431(CHEMBL3087715)
Affinity DataKi:  375nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494429(CHEMBL3087711)
Affinity DataKi:  438nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494423(CHEMBL3087717)
Affinity DataKi:  470nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494433(CHEMBL3087713)
Affinity DataKi:  496nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50256842(8-Bromo-9-methyl-9H-adenine | CHEMBL510288)
Affinity DataKi:  570nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494434(CHEMBL3087708)
Affinity DataKi:  583nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50257051(2-(6-amino-8-bromo-9H-purin-9-yl)ethanol | 8-Bromo...)
Affinity DataKi:  620nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494432(CHEMBL3087709)
Affinity DataKi:  652nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50256842(8-Bromo-9-methyl-9H-adenine | CHEMBL510288)
Affinity DataKi:  720nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494426(CHEMBL3087714)
Affinity DataKi:  756nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494430(CHEMBL3087716)
Affinity DataKi:  786nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494425(CHEMBL3087706)
Affinity DataKi:  790nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494424(CHEMBL3087710)
Affinity DataKi:  792nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50256890(8-Bromo-9-ethyl-9H-adenine | CHEMBL468633)
Affinity DataKi:  840nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494428(CHEMBL3087712)
Affinity DataKi:  906nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494428(CHEMBL3087712)
Affinity DataKi:  922nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50257054(8-Bromo-9-(3-hydroxypropyl)-9H-adenine | CHEMBL475...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50256893(8-Bromo-9-propyl-9H-adenine | CHEMBL506450)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494432(CHEMBL3087709)
Affinity DataKi:  1.27E+3nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50257051(2-(6-amino-8-bromo-9H-purin-9-yl)ethanol | 8-Bromo...)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494434(CHEMBL3087708)
Affinity DataKi:  1.95E+3nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494434(CHEMBL3087708)
Affinity DataKi:  2.51E+3nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494428(CHEMBL3087712)
Affinity DataKi:  2.78E+3nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50257051(2-(6-amino-8-bromo-9H-purin-9-yl)ethanol | 8-Bromo...)
Affinity DataKi:  2.80E+3nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50494424(CHEMBL3087710)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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