Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50043669
TargetProteasome subunit beta type-5(Homo sapiens (Human))
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50398608(MARIZOMIB)
Affinity DataIC50:  22nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome after 1 hr by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50444464(CHEMBL192046)
Affinity DataIC50:  23nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome after 1 hr by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50444462(CHEMBL3092609)
Affinity DataIC50:  28nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome after 1 hr by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50444463(CHEMBL3092608)
Affinity DataIC50:  50nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome after 1 hr by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50444466(CHEMBL3092611)
Affinity DataIC50:  330nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome after 1 hr by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50444461(CHEMBL3092610)
Affinity DataIC50:  500nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome after 1 hr by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50444465(CHEMBL3092612)
Affinity DataIC50:  500nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome after 1 hr by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50444464(CHEMBL192046)
Affinity DataEC50:  10nMAssay Description:Inhibition of chymotrypsin like activity of 20S proteasome in HEK293 cells after 24 hrs by microscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50444463(CHEMBL3092608)
Affinity DataEC50:  90nMAssay Description:Inhibition of chymotrypsin like activity of 20S proteasome in HEK293 cells after 24 hrs by microscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50444462(CHEMBL3092609)
Affinity DataEC50:  360nMAssay Description:Inhibition of chymotrypsin like activity of 20S proteasome in HEK293 cells after 24 hrs by microscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50444461(CHEMBL3092610)
Affinity DataEC50:  332nMAssay Description:Inhibition of chymotrypsin like activity of 20S proteasome in HEK293 cells after 24 hrs by microscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed