Compile Data Set for Download or QSAR
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Found 10 Enz. Inhib. hit(s) with all data for entry = 50044155
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50006650(CHEMBL526479)
Affinity DataIC50:  0.0300nMAssay Description:Inhibition of BRAF (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50006653(CHEMBL497671)
Affinity DataIC50:  0.220nMAssay Description:Inhibition of BRAF (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50006652(CHEMBL498674)
Affinity DataIC50:  0.340nMAssay Description:Inhibition of BRAF (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50432397(CHEMBL2348989)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50006650(CHEMBL526479)
Affinity DataIC50:  9nMAssay Description:Inhibition of BRAF (unknown origin)-mediated ERK phosphorylationMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50006651(CHEMBL3133758)
Affinity DataIC50:  22nMAssay Description:Inhibition of BRAF (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50432397(CHEMBL2348989)
Affinity DataIC50:  43nMAssay Description:Inhibition of BRAF (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50006651(CHEMBL3133758)
Affinity DataIC50:  95nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50006651(CHEMBL3133758)
Affinity DataIC50:  165nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50006649(CHEMBL3235904)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of N-terminal 6X-His tagged human wild-type BRAF by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed