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Found 14 Enz. Inhib. hit(s) with all data for entry = 50043874
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50447827(CHEMBL3114023)
Affinity DataIC50:  52nMAssay Description:Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM26474(5-({4-[(2,3-dimethyl-2H-indazol-6-yl)(methyl)amino...)
Affinity DataIC50:  71nMAssay Description:Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50447821(CHEMBL3114029)
Affinity DataIC50:  72nMAssay Description:Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50447820(CHEMBL3114030)
Affinity DataIC50:  75nMAssay Description:Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50447828(CHEMBL3114022)
Affinity DataIC50:  80nMAssay Description:Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50447830(CHEMBL3114020)
Affinity DataIC50:  85nMAssay Description:Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50447822(CHEMBL3114028)
Affinity DataIC50:  86nMAssay Description:Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50447826(CHEMBL3114024)
Affinity DataIC50:  94nMAssay Description:Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50447823(CHEMBL3114027)
Affinity DataIC50:  95nMAssay Description:Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50447829(CHEMBL3114021)
Affinity DataIC50:  96nMAssay Description:Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50447831(CHEMBL3114019)
Affinity DataIC50:  97nMAssay Description:Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50447825(CHEMBL3114025)
Affinity DataIC50:  104nMAssay Description:Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50447832(CHEMBL3114018)
Affinity DataIC50:  130nMAssay Description:Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50447824(CHEMBL3114026)
Affinity DataIC50:  140nMAssay Description:Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed