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Found 22 Enz. Inhib. hit(s) with all data for entry = 50043909
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Teva Pharmaceutical Global R & D

Curated by ChEMBL
LigandPNGBDBM50364958(CHEMBL1950743)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Teva Pharmaceutical Global R & D

Curated by ChEMBL
LigandPNGBDBM50448291(CHEMBL3121099)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Teva Pharmaceutical Global R & D

Curated by ChEMBL
LigandPNGBDBM50448285(CHEMBL3121093)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Teva Pharmaceutical Global R & D

Curated by ChEMBL
LigandPNGBDBM50448290(CHEMBL3121100)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Teva Pharmaceutical Global R & D

Curated by ChEMBL
LigandPNGBDBM50448293(CHEMBL3121097)
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Teva Pharmaceutical Global R & D

Curated by ChEMBL
LigandPNGBDBM50350021(CHEMBL1813067)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Teva Pharmaceutical Global R & D

Curated by ChEMBL
LigandPNGBDBM50448295(CHEMBL3121095)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Teva Pharmaceutical Global R & D

Curated by ChEMBL
LigandPNGBDBM50448292(CHEMBL3121098)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Teva Pharmaceutical Global R & D

Curated by ChEMBL
LigandPNGBDBM50448286(CHEMBL3121092)
Affinity DataKi:  8.10nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Teva Pharmaceutical Global R & D

Curated by ChEMBL
LigandPNGBDBM50448296(CHEMBL3121094)
Affinity DataKi:  8.40nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Teva Pharmaceutical Global R & D

Curated by ChEMBL
LigandPNGBDBM50448294(CHEMBL3121096)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Teva Pharmaceutical Global R & D

Curated by ChEMBL
LigandPNGBDBM50448287(CHEMBL3121091)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Teva Pharmaceutical Global R & D

Curated by ChEMBL
LigandPNGBDBM50448288(CHEMBL3121090)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Teva Pharmaceutical Global R & D

Curated by ChEMBL
LigandPNGBDBM50448289(CHEMBL3121101)
Affinity DataKi:  228nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Teva Pharmaceutical Global R & D

Curated by ChEMBL
LigandPNGBDBM50448294(CHEMBL3121096)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Teva Pharmaceutical Global R & D

Curated by ChEMBL
LigandPNGBDBM50448295(CHEMBL3121095)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Teva Pharmaceutical Global R & D

Curated by ChEMBL
LigandPNGBDBM50448294(CHEMBL3121096)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Teva Pharmaceutical Global R & D

Curated by ChEMBL
LigandPNGBDBM50448294(CHEMBL3121096)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Teva Pharmaceutical Global R & D

Curated by ChEMBL
LigandPNGBDBM50448294(CHEMBL3121096)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Teva Pharmaceutical Global R & D

Curated by ChEMBL
LigandPNGBDBM50448295(CHEMBL3121095)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Teva Pharmaceutical Global R & D

Curated by ChEMBL
LigandPNGBDBM50448295(CHEMBL3121095)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Teva Pharmaceutical Global R & D

Curated by ChEMBL
LigandPNGBDBM50448295(CHEMBL3121095)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed