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Found 20 Enz. Inhib. hit(s) with all data for entry = 50043967
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50449144(CHEMBL3127454)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using N14Y as substrate after 15 mins by PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50449148(CHEMBL3127450)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using N14Y as substrate after 15 mins by PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50449145(CHEMBL3127453)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using N14Y as substrate after 15 mins by PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50449159(CHEMBL3127439)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using N14Y as substrate after 15 mins by PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50449156(CHEMBL3127442)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using N14Y as substrate after 15 mins by PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50449153(CHEMBL3127445)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using N14Y as substrate after 15 mins by PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50449150(CHEMBL3127448)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using N14Y as substrate after 15 mins by PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50449147(CHEMBL3127451)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using N14Y as substrate after 15 mins by PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50449152(CHEMBL3127446)
Affinity DataIC50: >1.11E+5nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using N14Y as substrate after 15 mins by PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50449160(CHEMBL3127438)
Affinity DataIC50: >1.11E+5nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using N14Y as substrate after 15 mins by PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50449154(CHEMBL3127444)
Affinity DataIC50: >1.11E+5nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using N14Y as substrate after 15 mins by PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50449155(CHEMBL3127443)
Affinity DataIC50: >1.11E+5nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using N14Y as substrate after 15 mins by PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50449161(CHEMBL3127437)
Affinity DataIC50: >1.11E+5nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using N14Y as substrate after 15 mins by PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50449146(CHEMBL3127452)
Affinity DataIC50: >1.11E+5nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using N14Y as substrate after 15 mins by PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50449151(CHEMBL3127447)
Affinity DataIC50: >1.11E+5nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using N14Y as substrate after 15 mins by PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50449162(CHEMBL3127436)
Affinity DataIC50: >1.11E+5nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using N14Y as substrate after 15 mins by PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50449149(CHEMBL3127449)
Affinity DataIC50: >1.11E+5nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using N14Y as substrate after 15 mins by PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50449163(CHEMBL3127435)
Affinity DataIC50: >1.11E+5nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using N14Y as substrate after 15 mins by PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50449158(CHEMBL3127440)
Affinity DataIC50: >1.11E+5nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using N14Y as substrate after 15 mins by PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50449157(CHEMBL3127441)
Affinity DataIC50: >1.11E+5nMAssay Description:Inhibition of recombinant TDP1 (unknown origin) using N14Y as substrate after 15 mins by PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed