Found 20 Enz. Inhib. hit(s) with all data for entry = 50044457 TargetRAS guanyl-releasing protein 1(Homo sapiens (Human))
National Institute Of Industrial Technology
Curated by ChEMBL
National Institute Of Industrial Technology
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H]PDBu from recombinant RasGRP1 C1 domain (unknown origin) after 10 mins by scintillation counting analysis in presence of phosphat...More data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Institute Of Industrial Technology
Curated by ChEMBL
National Institute Of Industrial Technology
Curated by ChEMBL
Affinity DataKi: 0.330nMAssay Description:Displacement of [3H]PDBu from recombinant human GFP-tagged RasGRP3 expressed in Escherichia coli BL21 after 5 mins by scintillation counting analysis...More data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Institute Of Industrial Technology
Curated by ChEMBL
National Institute Of Industrial Technology
Curated by ChEMBL
Affinity DataKi: 0.340nMAssay Description:Displacement of [3H]PDBu from recombinant human GFP-tagged RasGRP3 expressed in Escherichia coli BL21 after 5 mins by scintillation counting analysis...More data for this Ligand-Target Pair
TargetRAS guanyl-releasing protein 1(Homo sapiens (Human))
National Institute Of Industrial Technology
Curated by ChEMBL
National Institute Of Industrial Technology
Curated by ChEMBL
Affinity DataKi: 0.410nMAssay Description:Displacement of [3H]PDBu from recombinant RasGRP1 C1 domain (unknown origin) after 10 mins by scintillation counting analysis in presence of phosphat...More data for this Ligand-Target Pair
TargetRAS guanyl-releasing protein 1(Homo sapiens (Human))
National Institute Of Industrial Technology
Curated by ChEMBL
National Institute Of Industrial Technology
Curated by ChEMBL
Affinity DataKi: 0.690nMAssay Description:Displacement of [3H]PDBu from recombinant RasGRP1 C1 domain (unknown origin) after 10 mins by scintillation counting analysis in presence of phosphat...More data for this Ligand-Target Pair
TargetRAS guanyl-releasing protein 1(Homo sapiens (Human))
National Institute Of Industrial Technology
Curated by ChEMBL
National Institute Of Industrial Technology
Curated by ChEMBL
Affinity DataKi: 0.870nMAssay Description:Displacement of [3H]PDBu from recombinant RasGRP1 C1 domain (unknown origin) after 10 mins by scintillation counting analysis in presence of phosphat...More data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Institute Of Industrial Technology
Curated by ChEMBL
National Institute Of Industrial Technology
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]PDBu from recombinant human GFP-tagged RasGRP3 expressed in Escherichia coli BL21 after 5 mins by scintillation counting analysis...More data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Institute Of Industrial Technology
Curated by ChEMBL
National Institute Of Industrial Technology
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]PDBu from recombinant human GFP-tagged RasGRP3 expressed in Escherichia coli BL21 after 5 mins by scintillation counting analysis...More data for this Ligand-Target Pair
TargetRAS guanyl-releasing protein 1(Homo sapiens (Human))
National Institute Of Industrial Technology
Curated by ChEMBL
National Institute Of Industrial Technology
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]PDBu from recombinant RasGRP1 C1 domain (unknown origin) after 10 mins by scintillation counting analysis in presence of phosphat...More data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Institute Of Industrial Technology
Curated by ChEMBL
National Institute Of Industrial Technology
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]PDBu from recombinant human GFP-tagged RasGRP3 expressed in Escherichia coli BL21 after 5 mins by scintillation counting analysis...More data for this Ligand-Target Pair
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute Of Industrial Technology
Curated by ChEMBL
National Institute Of Industrial Technology
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-epsilon after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Institute Of Industrial Technology
Curated by ChEMBL
National Institute Of Industrial Technology
Curated by ChEMBL
Affinity DataKi: 7.5nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-alpha after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute Of Industrial Technology
Curated by ChEMBL
National Institute Of Industrial Technology
Curated by ChEMBL
Affinity DataKi: 8.10nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-epsilon after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Institute Of Industrial Technology
Curated by ChEMBL
National Institute Of Industrial Technology
Curated by ChEMBL
Affinity DataKi: 8.30nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-alpha after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute Of Industrial Technology
Curated by ChEMBL
National Institute Of Industrial Technology
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-epsilon after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Institute Of Industrial Technology
Curated by ChEMBL
National Institute Of Industrial Technology
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-alpha after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute Of Industrial Technology
Curated by ChEMBL
National Institute Of Industrial Technology
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-epsilon after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Institute Of Industrial Technology
Curated by ChEMBL
National Institute Of Industrial Technology
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-alpha after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Institute Of Industrial Technology
Curated by ChEMBL
National Institute Of Industrial Technology
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-alpha after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute Of Industrial Technology
Curated by ChEMBL
National Institute Of Industrial Technology
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-epsilon after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
