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Found 38 Enz. Inhib. hit(s) with all data for entry = 50044599
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021819(CHEMBL3298828)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021818(CHEMBL3298827)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021817(CHEMBL3298826)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021771(CHEMBL3298896)
Affinity DataKi:  9.10nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021770(CHEMBL3298895)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021802(CHEMBL3299096)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021769(CHEMBL3298830)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021796(CHEMBL3299094)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021800(CHEMBL3299095)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021816(CHEMBL3298759)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021768(CHEMBL3298829)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021815(CHEMBL3298758)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021805(CHEMBL3299097)
Affinity DataKi:  75nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021791(CHEMBL3299093)
Affinity DataKi:  170nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021789(CHEMBL3299092)
Affinity DataKi:  902nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021806(CHEMBL3299098)
Affinity DataKi:  910nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021814(CHEMBL3298686)
Affinity DataKi:  975nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50394930(CHEMBL1424807)
Affinity DataKi:  1.16E+3nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021774(CHEMBL3298757)
Affinity DataKi:  1.35E+3nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021810(CHEMBL3299099)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021813(CHEMBL3298685)
Affinity DataKi:  1.98E+3nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021788(CHEMBL3299091)
Affinity DataKi:  2.05E+3nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021775(CHEMBL3298825)
Affinity DataKi:  2.11E+3nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021811(CHEMBL3298200)
Affinity DataKi:  2.25E+3nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021773(CHEMBL3298756)
Affinity DataKi:  2.75E+3nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50001862((N-(o-methoxyphenyl)piperazine)1-(2-Methoxy-phenyl...)
Affinity DataKi:  4.11E+3nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021772(CHEMBL3298755 | EN300-127205)
Affinity DataKi:  9.09E+3nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in FlpIn CHO cell membrane after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021805(CHEMBL3299097)
Affinity DataIC50:  4nMAssay Description:Antagonist activity at human D2L receptor expressed in FlpIn CHO cells assessed as inhibition of dopamine-induced ERK1/2 phosphorylation treated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021791(CHEMBL3299093)
Affinity DataIC50:  93nMAssay Description:Antagonist activity at human D2L receptor expressed in FlpIn CHO cells assessed as inhibition of dopamine-induced ERK1/2 phosphorylation treated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50001862((N-(o-methoxyphenyl)piperazine)1-(2-Methoxy-phenyl...)
Affinity DataIC50: >1.00E+3nMAssay Description:Antagonist activity at human D2L receptor expressed in FlpIn CHO cells assessed as inhibition of dopamine-induced ERK1/2 phosphorylation treated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021818(CHEMBL3298827)
Affinity DataEC50:  2.70nMAssay Description:Partial agonist activity at human D2L receptor expressed in FlpIn CHO cells assessed as induction of ERK1/2 phosphorylation by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021802(CHEMBL3299096)
Affinity DataEC50:  1.40nMAssay Description:Partial agonist activity at human D2L receptor expressed in FlpIn CHO cells assessed as induction of ERK1/2 phosphorylation by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021800(CHEMBL3299095)
Affinity DataEC50:  0.600nMAssay Description:Partial agonist activity at human D2L receptor expressed in FlpIn CHO cells assessed as induction of ERK1/2 phosphorylation by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021796(CHEMBL3299094)
Affinity DataEC50:  0.390nMAssay Description:Partial agonist activity at human D2L receptor expressed in FlpIn CHO cells assessed as induction of ERK1/2 phosphorylation by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021769(CHEMBL3298830)
Affinity DataEC50:  88nMAssay Description:Agonist activity at human D2L receptor expressed in FlpIn CHO cells assessed as induction of ERK1/2 phosphorylation by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021770(CHEMBL3298895)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at human D2L receptor expressed in FlpIn CHO cells assessed as inhibition of forskolin-stimulated cAMP production treated for 30 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021819(CHEMBL3298828)
Affinity DataEC50:  5.5nMAssay Description:Partial agonist activity at human D2L receptor expressed in FlpIn CHO cells assessed as induction of ERK1/2 phosphorylation by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50021770(CHEMBL3298895)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human D2L receptor expressed in FlpIn CHO cells assessed as induction of ERK1/2 phosphorylation by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed