Compile Data Set for Download or QSAR
maximum 50k data
Found 27 Enz. Inhib. hit(s) with all data for entry = 50039496
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379081(Aigialomycin D | CHEMBL1173442)
Affinity DataIC50:  450nMAssay Description:Inhibition of MNK2 using 5-FAM-TATKSGSTTKNRFVV-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 2 hrs by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379075(CHEMBL2012392)
Affinity DataIC50:  580nMAssay Description:Inhibition of MNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379073(CHEMBL2012390)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of MNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379083(CHEMBL2012384)
Affinity DataIC50:  1.61E+3nMAssay Description:Inhibition of MNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379081(Aigialomycin D | CHEMBL1173442)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of CDK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379081(Aigialomycin D | CHEMBL1173442)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of CDK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379074(CHEMBL2012389)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379072(CHEMBL2012387)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379071(CHEMBL2012386)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379070(CHEMBL2012388)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379078(CHEMBL2012394)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379085(CHEMBL2012382)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379084(CHEMBL2012383)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379082(CHEMBL2012385)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379080(CHEMBL2012396)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379079(CHEMBL2012395)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379077(CHEMBL2012393)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379076(CHEMBL2012391)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379078(CHEMBL2012394)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of CDK2/cyclin A using 5-FAM-GGGPATPKKAKKL-COOH as substrate after 1 hr by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379085(CHEMBL2012382)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of CDK2/cyclin A using 5-FAM-GGGPATPKKAKKL-COOH as substrate after 1 hr by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379081(Aigialomycin D | CHEMBL1173442)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of CDK2/cyclin A using 5-FAM-GGGPATPKKAKKL-COOH as substrate after 1 hr by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379081(Aigialomycin D | CHEMBL1173442)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of MNK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379081(Aigialomycin D | CHEMBL1173442)
Affinity DataKd:  1.20E+4nMAssay Description:Inhibition of PRKCEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379081(Aigialomycin D | CHEMBL1173442)
Affinity DataKd:  300nMAssay Description:Inhibition of FLT3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379081(Aigialomycin D | CHEMBL1173442)
Affinity DataKd:  1.00E+3nMAssay Description:Inhibition of AXLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379081(Aigialomycin D | CHEMBL1173442)
Affinity DataKd:  260nMAssay Description:Inhibition of PLK4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379081(Aigialomycin D | CHEMBL1173442)
Affinity DataKd:  160nMAssay Description:Inhibition of MNK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed