Compile Data Set for Download or QSAR
maximum 50k data
Found 51 Enz. Inhib. hit(s) with all data for entry = 50039813
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384652(CHEMBL2037112)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384653(CHEMBL2037113)
Affinity DataIC50:  5nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384650(CHEMBL2037096)
Affinity DataIC50:  5nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384648(CHEMBL2037114)
Affinity DataIC50:  7nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384654(CHEMBL2037018)
Affinity DataIC50:  14nMAssay Description:Competitive inhibition of CHK1 using ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384679(CHEMBL2037097)
Affinity DataIC50:  19nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384651(CHEMBL2037111)
Affinity DataIC50:  19nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384684(CHEMBL2037102)
Affinity DataIC50:  36nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384657(CHEMBL2037115)
Affinity DataIC50:  69nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384675(CHEMBL2037093)
Affinity DataIC50:  72nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384649(CHEMBL2037017)
Affinity DataIC50:  75nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384667(CHEMBL2037025)
Affinity DataIC50:  86nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384674(CHEMBL2037092)
Affinity DataIC50:  87nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384686(CHEMBL2037104)
Affinity DataIC50:  89nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384681(CHEMBL2037099)
Affinity DataIC50:  100nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384687(CHEMBL2037105)
Affinity DataIC50:  110nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384666(CHEMBL2037024)
Affinity DataIC50:  120nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384685(CHEMBL2037103)
Affinity DataIC50:  130nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384678(CHEMBL2037094)
Affinity DataIC50:  170nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384660(CHEMBL2037095)
Affinity DataIC50:  190nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384688(CHEMBL2037106)
Affinity DataIC50:  190nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384683(CHEMBL2037101)
Affinity DataIC50:  210nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384649(CHEMBL2037017)
Affinity DataIC50:  210nMAssay Description:Inhibition of Cyclin E/CDK2 expressed in Sf9 cells using [33gamma]ATP after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384663(CHEMBL2037021)
Affinity DataIC50:  280nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384658(CHEMBL2037116)
Affinity DataIC50:  440nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384677(CHEMBL2037085)
Affinity DataIC50:  520nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384676(CHEMBL2037084)
Affinity DataIC50:  580nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384662(CHEMBL2037020)
Affinity DataIC50:  760nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384682(CHEMBL2037100)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384690(CHEMBL2037108)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384689(CHEMBL2037107)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384668(CHEMBL2037086)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384673(CHEMBL2037091)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384659(CHEMBL2037117)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384669(CHEMBL2037087)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384661(CHEMBL2037019)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384655(CHEMBL2037109)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384656(CHEMBL2037110)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384671(CHEMBL2037089)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384680(CHEMBL2037098)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384670(CHEMBL2037088)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384672(CHEMBL2037090)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384664(CHEMBL2037022)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384665(CHEMBL2037023)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant His-tagged CHK1 using biotin-RSGLYRSPSMPENLNRPR as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384649(CHEMBL2037017)
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of CHK1 in human U2OS cells pretreated with hydroxyurea assessed as gamma-H2AX level after 2 hrs by immunofluorescence assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384651(CHEMBL2037111)
Affinity DataEC50:  2.00E+3nMAssay Description:Inhibition of CHK1 in human U2OS cells pretreated with hydroxyurea assessed as gamma-H2AX level after 2 hrs by immunofluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384649(CHEMBL2037017)
Affinity DataKd: <100nMAssay Description:Binding affinity to CHK1 by affinity-selection-mass spectrophotometry assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384650(CHEMBL2037096)
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of CHK1 in human U2OS cells pretreated with hydroxyurea assessed as gamma-H2AX level after 2 hrs by immunofluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384652(CHEMBL2037112)
Affinity DataEC50:  3.50E+3nMAssay Description:Inhibition of CHK1 in human U2OS cells pretreated with hydroxyurea assessed as gamma-H2AX level after 2 hrs by immunofluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384653(CHEMBL2037113)
Affinity DataEC50:  2.50E+3nMAssay Description:Inhibition of CHK1 in human U2OS cells pretreated with hydroxyurea assessed as gamma-H2AX level after 2 hrs by immunofluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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