Compile Data Set for Download or QSAR
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Found 13 Enz. Inhib. hit(s) with all data for entry = 50040077
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388923(CHEMBL2063283)
Affinity DataIC50:  28nMAssay Description:Inhibition of human recombinant His6-tagged DGAT1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388921(CHEMBL2063281)
Affinity DataIC50:  28nMAssay Description:Inhibition of human recombinant His6-tagged DGAT1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388924(CHEMBL2063284)
Affinity DataIC50:  39nMAssay Description:Inhibition of human recombinant His6-tagged DGAT1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388922(CHEMBL2063282)
Affinity DataIC50:  56nMAssay Description:Inhibition of human recombinant His6-tagged DGAT1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Mus musculus (mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50388920(CHEMBL2063280)
Affinity DataIC50:  120nMAssay Description:Inhibition of DGAT1 in mouse C2C12 cells assessed as reduction in triglyceride synthesis after 2 hrs by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Mus musculus (mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50388924(CHEMBL2063284)
Affinity DataIC50:  390nMAssay Description:Inhibition of DGAT1 in mouse C2C12 cells assessed as reduction in triglyceride synthesis after 2 hrs by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388920(CHEMBL2063280)
Affinity DataIC50:  500nMAssay Description:Inhibition of human recombinant His6-tagged DGAT1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388918(CHEMBL2063278)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human recombinant His6-tagged DGAT1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388919(CHEMBL2063279)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human recombinant His6-tagged DGAT1 expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Mus musculus (mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50388922(CHEMBL2063282)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of DGAT1 in mouse C2C12 cells assessed as reduction in triglyceride synthesis after 2 hrs by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Mus musculus (mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50388923(CHEMBL2063283)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of DGAT1 in mouse C2C12 cells assessed as reduction in triglyceride synthesis after 2 hrs by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Mus musculus (mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50388921(CHEMBL2063281)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of DGAT1 in mouse C2C12 cells assessed as reduction in triglyceride synthesis after 2 hrs by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388918(CHEMBL2063278)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of DGAT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed