Compile Data Set for Download or QSAR
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Found 8 Enz. Inhib. hit(s) with all data for entry = 50039692
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50382408(CHEMBL2022554)
Affinity DataIC50:  6.10E+3nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium accu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50382406(CHEMBL1606364)
Affinity DataIC50:  9.80E+3nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium accu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50382405(CHEMBL2022172)
Affinity DataIC50:  1.44E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium accu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50382406(CHEMBL1606364)
Affinity DataIC50:  1.96E+4nMAssay Description:Antagonist activity at human alpha3beta4 nAChR expressed in HEK tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium accu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50382407(CHEMBL1536503)
Affinity DataIC50:  2.06E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium accu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50382405(CHEMBL2022172)
Affinity DataIC50:  4.63E+4nMAssay Description:Antagonist activity at human alpha3beta4 nAChR expressed in HEK tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium accu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50382407(CHEMBL1536503)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human alpha3beta4 nAChR expressed in HEK tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium accu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50382408(CHEMBL2022554)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human alpha3beta4 nAChR expressed in HEK tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium accu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed