Affinity DataKi: 1.01E+3nMAssay Description:Inhibition of DAT (unknown origin)-mediated dopamine reuptakeMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataIC50: 294nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataIC50: 369nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataIC50: 386nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataIC50: 425nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataIC50: 533nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataIC50: 592nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataIC50: 793nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataIC50: 2.01E+3nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataIC50: 2.37E+3nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataIC50: 3.18E+3nMAssay Description:Inhibition of SERT-mediated serotonin uptake in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataIC50: 5.92E+3nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SERT-mediated serotonin uptake in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SERT-mediated serotonin uptake in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SERT-mediated serotonin uptake in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SERT-mediated serotonin uptake in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataEC50: 2.12E+3nMAssay Description:Induction of SERT (unknown origin)-mediated serotonin releaseMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataEC50: 181nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataEC50: 410nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataEC50: 4.70E+3nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataEC50: 1.33E+3nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataEC50: 562nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataEC50: 733nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataEC50: 621nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataEC50: 1.07E+3nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataEC50: 1.01E+3nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataEC50: 1.63E+3nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataEC50: 356nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataEC50: 667nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataEC50: 411nMAssay Description:Induction of DAT-mediated dopamine release in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataEC50: 225nMAssay Description:Induction of DAT-mediated dopamine release in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Induction of DAT-mediated dopamine release in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataEC50: 47nMAssay Description:Induction of DAT-mediated dopamine release in rat synaptosomesMore data for this Ligand-Target Pair