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Found 7 Enz. Inhib. hit(s) with all data for entry = 50045303
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50055958(CHEMBL3326555)
Affinity DataIC50:  20nMAssay Description:Inhibition of full-length human PIM3 using RSRHSSYPAGT as substrate assessed as residual kinase activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50055958(CHEMBL3326555)
Affinity DataIC50:  70nMAssay Description:Inhibition of full-length human PIM1 using RSRHSSYPAGT as substrate assessed as residual kinase activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50055959(CHEMBL3326556)
Affinity DataIC50:  120nMAssay Description:Inhibition of full-length human PIM1 using RSRHSSYPAGT as substrate assessed as residual kinase activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50055959(CHEMBL3326556)
Affinity DataIC50:  140nMAssay Description:Inhibition of full-length human PIM3 using RSRHSSYPAGT as substrate assessed as residual kinase activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50055961(CHEMBL3326558)
Affinity DataIC50:  169nMAssay Description:Inhibition of full-length human PIM3 using RSRHSSYPAGT as substrate assessed as residual kinase activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50055960(CHEMBL3326557)
Affinity DataIC50:  200nMAssay Description:Inhibition of full-length human PIM3 using RSRHSSYPAGT as substrate assessed as residual kinase activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50055962(CHEMBL3326559)
Affinity DataIC50:  400nMAssay Description:Inhibition of full-length human PIM3 using RSRHSSYPAGT as substrate assessed as residual kinase activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed