TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 2.40E+3nMAssay Description:Displacement of [3H] CP-55,940 from human CB2 receptor expressed in HEK cells at 10 uM after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 1.27E+4nMAssay Description:Displacement of [3H] CP-55,940 from human CB2 receptor expressed in HEK cells at 10 uM after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 3.10E+4nMAssay Description:Displacement of [3H] CP-55,940 from human CB2 receptor expressed in HEK cells at 10 uM after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 1.35E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 1.50E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 4.07E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 9.55E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 9.66E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 8.71E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 8.55E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 7.60E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 2.43E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 3.16E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 1.05E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 1.62E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 7.24E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 8.85E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 2.95E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 776nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 501nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 110nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 1.10E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 661nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 123nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 1.62E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 1.91E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 68nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 50nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 2.82E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 112nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 3.89E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 871nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 1.35E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 1.51E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 4.07E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 9.55E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 9.55E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 8.71E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 8.51E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 7.59E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 2.40E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 3.16E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 1.05E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 1.62E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 7.24E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 8.91E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 2.95E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 776nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 501nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 110nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair