Compile Data Set for Download or QSAR
maximum 50k data
Found 63 Enz. Inhib. hit(s) with all data for entry = 50045314
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056333(CHEMBL3322470)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [3H] CP-55,940 from human CB2 receptor expressed in HEK cells at 10 uM after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056338(CHEMBL3322475)
Affinity DataKi:  1.27E+4nMAssay Description:Displacement of [3H] CP-55,940 from human CB2 receptor expressed in HEK cells at 10 uM after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056339(CHEMBL3322476)
Affinity DataKi:  3.10E+4nMAssay Description:Displacement of [3H] CP-55,940 from human CB2 receptor expressed in HEK cells at 10 uM after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056319(CHEMBL3322458)
Affinity DataEC50:  1.35E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056320(CHEMBL3322454)
Affinity DataEC50:  1.50E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056321(CHEMBL3322455)
Affinity DataEC50:  4.07E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056322(CHEMBL3322457)
Affinity DataEC50:  9.55E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056323(CHEMBL3322459)
Affinity DataEC50:  9.66E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056324(CHEMBL3322460)
Affinity DataEC50:  8.71E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056325(CHEMBL3322461)
Affinity DataEC50:  8.55E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056326(CHEMBL3322462)
Affinity DataEC50:  7.60E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056327(CHEMBL3322463)
Affinity DataEC50:  2.43E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056328(CHEMBL3322464)
Affinity DataEC50:  3.16E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056329(CHEMBL3322465)
Affinity DataEC50:  1.05E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056330(CHEMBL3322467)
Affinity DataEC50:  1.62E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056331(CHEMBL3322468)
Affinity DataEC50:  7.24E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056332(CHEMBL3322469)
Affinity DataEC50:  8.85E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056333(CHEMBL3322470)
Affinity DataEC50:  2.95E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056334(CHEMBL3322471)
Affinity DataEC50:  776nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056335(CHEMBL3322472)
Affinity DataEC50:  501nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056336(CHEMBL3322473)
Affinity DataEC50:  110nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056337(CHEMBL3322474)
Affinity DataEC50:  1.10E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056338(CHEMBL3322475)
Affinity DataEC50:  661nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056339(CHEMBL3322476)
Affinity DataEC50:  123nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056340(CHEMBL3322478)
Affinity DataEC50:  1.62E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056341(CHEMBL3322479)
Affinity DataEC50:  1.91E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM21279(1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N...)
Affinity DataEC50:  68nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataEC50:  50nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056316(CHEMBL3322348)
Affinity DataEC50:  2.82E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056317(CHEMBL3322349)
Affinity DataEC50:  112nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056318(CHEMBL3322350)
Affinity DataEC50:  3.89E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50328952(CHEMBL1269766 | N,N'-(Iminodiheptane-7,1-diyl)bis[...)
Affinity DataEC50:  871nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056319(CHEMBL3322458)
Affinity DataEC50:  1.35E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056320(CHEMBL3322454)
Affinity DataEC50:  1.51E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056321(CHEMBL3322455)
Affinity DataEC50:  4.07E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056322(CHEMBL3322457)
Affinity DataEC50:  9.55E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056323(CHEMBL3322459)
Affinity DataEC50:  9.55E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056324(CHEMBL3322460)
Affinity DataEC50:  8.71E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056325(CHEMBL3322461)
Affinity DataEC50:  8.51E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056326(CHEMBL3322462)
Affinity DataEC50:  7.59E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056327(CHEMBL3322463)
Affinity DataEC50:  2.40E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056328(CHEMBL3322464)
Affinity DataEC50:  3.16E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056329(CHEMBL3322465)
Affinity DataEC50:  1.05E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056330(CHEMBL3322467)
Affinity DataEC50:  1.62E+4nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056331(CHEMBL3322468)
Affinity DataEC50:  7.24E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056332(CHEMBL3322469)
Affinity DataEC50:  8.91E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056333(CHEMBL3322470)
Affinity DataEC50:  2.95E+3nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056334(CHEMBL3322471)
Affinity DataEC50:  776nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056335(CHEMBL3322472)
Affinity DataEC50:  501nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056336(CHEMBL3322473)
Affinity DataEC50:  110nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in Sf9 cells coexpressing Gbeta1gamma2 and RSG4 assessed as degradation of [gamma-33P]GTP af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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