Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with all data for entry = 6833
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

LigandPNGBDBM15211(CHEMBL104264 | H-89 | H89 | HT-89 (H-89) | N-(2-{[...)
Affinity DataIC50:  1.70E+3nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assays were carried out using HTScanŽ PKB/Akt1 Kinase Assay kit (Cell Signaling Technology). Active recombinant Akt1 kinase (GST fusi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

LigandPNGBDBM153374(6-((Benzyl(methyl)amino)methyl)-2-(3,4-dihydroxyph...)
Affinity DataIC50:  5.50E+3nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assays were carried out using HTScanŽ PKB/Akt1 Kinase Assay kit (Cell Signaling Technology). Active recombinant Akt1 kinase (GST fusi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

LigandPNGBDBM153373(2-(3,4-Dihydroxyphenyl)-3,5,7-trihydroxy-6-(morpho...)
Affinity DataIC50:  6.20E+3nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assays were carried out using HTScanŽ PKB/Akt1 Kinase Assay kit (Cell Signaling Technology). Active recombinant Akt1 kinase (GST fusi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed