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Found 21 Enz. Inhib. hit(s) with all data for entry = 50044912
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University

Curated by ChEMBL
LigandPNGBDBM50059863((Z)-2-Methyl-3-tetradecyl-but-2-enedioic acid | CH...)
Affinity DataIC50:  180nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University

Curated by ChEMBL
LigandPNGBDBM50036274(CHEMBL3361086)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University

Curated by ChEMBL
LigandPNGBDBM50036270(CHEMBL3361094)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University

Curated by ChEMBL
LigandPNGBDBM50035931(CHEMBL3361085)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University

Curated by ChEMBL
LigandPNGBDBM50036277(CHEMBL3361077)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University

Curated by ChEMBL
LigandPNGBDBM50036276(CHEMBL3361076)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University

Curated by ChEMBL
LigandPNGBDBM50036272(CHEMBL3361092)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University

Curated by ChEMBL
LigandPNGBDBM50035927(CHEMBL3361080)
Affinity DataIC50:  1.14E+4nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University

Curated by ChEMBL
LigandPNGBDBM50035929(CHEMBL3361082)
Affinity DataIC50:  1.44E+4nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University

Curated by ChEMBL
LigandPNGBDBM50035921(CHEMBL3361071)
Affinity DataIC50:  1.48E+4nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University

Curated by ChEMBL
LigandPNGBDBM50035926(CHEMBL3361079)
Affinity DataIC50:  1.49E+4nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University

Curated by ChEMBL
LigandPNGBDBM50035928(CHEMBL3361081)
Affinity DataIC50:  1.53E+4nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University

Curated by ChEMBL
LigandPNGBDBM50035923(CHEMBL3361068)
Affinity DataIC50:  1.94E+4nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University

Curated by ChEMBL
LigandPNGBDBM50035925(CHEMBL3361066)
Affinity DataIC50:  1.97E+4nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University

Curated by ChEMBL
LigandPNGBDBM50035924(CHEMBL3361067)
Affinity DataIC50:  2.07E+4nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University

Curated by ChEMBL
LigandPNGBDBM50036273(CHEMBL3361093)
Affinity DataIC50:  2.07E+4nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University

Curated by ChEMBL
LigandPNGBDBM50035930(CHEMBL3361084)
Affinity DataIC50:  2.08E+4nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University

Curated by ChEMBL
LigandPNGBDBM50036275(CHEMBL3361075)
Affinity DataIC50:  2.21E+4nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University

Curated by ChEMBL
LigandPNGBDBM50035922(CHEMBL3361070)
Affinity DataIC50:  3.22E+4nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University

Curated by ChEMBL
LigandPNGBDBM50036278(CHEMBL3361078)
Affinity DataIC50:  5.78E+4nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University

Curated by ChEMBL
LigandPNGBDBM50036271(CHEMBL3361072)
Affinity DataIC50:  7.23E+4nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed