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Found 4 Enz. Inhib. hit(s) with all data for entry = 50044927
TargetAcetylcholinesterase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  20nMAssay Description:Inhibition of AChE (unknown origin) assessed as inhibition of acetylcholine hydrolysis preincubated for 15 mins by Ellman methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50036515(CHEMBL3353567)
Affinity DataIC50:  5.30E+4nMAssay Description:Inhibition of AChE (unknown origin) assessed as inhibition of acetylcholine hydrolysis preincubated for 15 mins by Ellman methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50036514(CHEMBL3353566)
Affinity DataIC50:  6.30E+4nMAssay Description:Inhibition of AChE (unknown origin) assessed as inhibition of acetylcholine hydrolysis preincubated for 15 mins by Ellman methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50036516(CHEMBL3353568)
Affinity DataIC50:  6.80E+4nMAssay Description:Inhibition of AChE (unknown origin) assessed as inhibition of acetylcholine hydrolysis preincubated for 15 mins by Ellman methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed