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Found 17 Enz. Inhib. hit(s) with all data for entry = 50045993
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50089907(CHEMBL3581056)
Affinity DataKi:  440nMAssay Description:Inhibition of Nav1.7 (unknown origin) by electrophysiological assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50089904(CHEMBL3581058)
Affinity DataKi:  560nMAssay Description:Inhibition of Nav1.7 (unknown origin) by electrophysiological assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50089917(CHEMBL3581050)
Affinity DataKi:  650nMAssay Description:Inhibition of Nav1.7 (unknown origin) by electrophysiological assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50089918(CHEMBL3581059)
Affinity DataKi:  920nMAssay Description:Inhibition of Nav1.7 (unknown origin) by electrophysiological assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50089908(CHEMBL3581054)
Affinity DataKi:  1.03E+3nMAssay Description:Inhibition of Nav1.7 (unknown origin) by electrophysiological assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50089915(CHEMBL3581053)
Affinity DataKi:  3.03E+3nMAssay Description:Inhibition of Nav1.7 (unknown origin) by electrophysiological assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50003659(5H-dibenzo[b,f]azepine-5-carboxamide | CARBAMAZEPI...)
Affinity DataKi:  3.27E+4nMAssay Description:Inhibition of Nav1.7 (unknown origin) by electrophysiological assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50089907(CHEMBL3581056)
Affinity DataIC50:  370nMAssay Description:Inhibition of Nav1.7 (unknown origin) expressed in CHO cells after 45 mins by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50089922(CHEMBL3581051)
Affinity DataIC50:  840nMAssay Description:Inhibition of Nav1.7 (unknown origin) expressed in CHO cells after 45 mins by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50089904(CHEMBL3581058)
Affinity DataIC50:  1.03E+3nMAssay Description:Inhibition of Nav1.7 (unknown origin) expressed in CHO cells after 45 mins by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50089918(CHEMBL3581059)
Affinity DataIC50:  1.05E+3nMAssay Description:Inhibition of Nav1.7 (unknown origin) expressed in CHO cells after 45 mins by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50089908(CHEMBL3581054)
Affinity DataIC50:  1.08E+3nMAssay Description:Inhibition of Nav1.7 (unknown origin) expressed in CHO cells after 45 mins by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50089919(CHEMBL3581057)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of Nav1.7 (unknown origin) expressed in CHO cells after 45 mins by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50089917(CHEMBL3581050)
Affinity DataIC50:  1.96E+3nMAssay Description:Inhibition of Nav1.7 (unknown origin) expressed in CHO cells after 45 mins by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50089920(CHEMBL3581055)
Affinity DataIC50:  2.57E+3nMAssay Description:Inhibition of Nav1.7 (unknown origin) expressed in CHO cells after 45 mins by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50089915(CHEMBL3581053)
Affinity DataIC50:  7.62E+3nMAssay Description:Inhibition of Nav1.7 (unknown origin) expressed in CHO cells after 45 mins by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50089921(CHEMBL3581052)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Nav1.7 (unknown origin) expressed in CHO cells after 45 mins by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed