Compile Data Set for Download or QSAR
maximum 50k data
Found 34 Enz. Inhib. hit(s) with all data for entry = 50045957
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088564(CHEMBL3577041)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM15581(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088560(CHEMBL3577045)
Affinity DataIC50:  18nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088568(CHEMBL3577037)
Affinity DataIC50:  33nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088563(CHEMBL3577042)
Affinity DataIC50:  36nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088565(CHEMBL3577040)
Affinity DataIC50:  36nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088562(CHEMBL3577043)
Affinity DataIC50:  43nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088557(CHEMBL3577048)
Affinity DataIC50:  48nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088559(CHEMBL3577046)
Affinity DataIC50:  49nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM22787(1-acetyl-2,3-dihydro-1H-indole-2,3-dione | Acetyli...)
Affinity DataIC50:  56nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088554(CHEMBL3577036)
Affinity DataIC50:  58nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088561(CHEMBL3577044)
Affinity DataIC50:  60nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088567(CHEMBL3577038)
Affinity DataIC50:  62nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088566(CHEMBL3577039)
Affinity DataIC50:  68nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088555(CHEMBL3577035)
Affinity DataIC50:  72nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088556(CHEMBL3577034)
Affinity DataIC50:  83nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
King Saud University

Curated by ChEMBL
LigandPNGBDBM15581(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Affinity DataIC50:  9.80E+4nMAssay Description:Inhibition of MAO-B in bovine brain mitochondria using benzylamine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088563(CHEMBL3577042)
Affinity DataIC50:  2.80E+5nMAssay Description:Inhibition of MAO-B in bovine brain mitochondria using benzylamine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088562(CHEMBL3577043)
Affinity DataIC50:  3.60E+5nMAssay Description:Inhibition of MAO-B in bovine brain mitochondria using benzylamine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
King Saud University

Curated by ChEMBL
LigandPNGBDBM22787(1-acetyl-2,3-dihydro-1H-indole-2,3-dione | Acetyli...)
Affinity DataIC50:  3.80E+5nMAssay Description:Inhibition of MAO-B in bovine brain mitochondria using benzylamine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088557(CHEMBL3577048)
Affinity DataIC50:  3.80E+5nMAssay Description:Inhibition of MAO-B in bovine brain mitochondria using benzylamine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088564(CHEMBL3577041)
Affinity DataIC50:  4.30E+5nMAssay Description:Inhibition of MAO-B in bovine brain mitochondria using benzylamine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088554(CHEMBL3577036)
Affinity DataIC50:  4.59E+5nMAssay Description:Inhibition of MAO-B in bovine brain mitochondria using benzylamine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088555(CHEMBL3577035)
Affinity DataIC50:  4.80E+5nMAssay Description:Inhibition of MAO-B in bovine brain mitochondria using benzylamine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088560(CHEMBL3577045)
Affinity DataIC50:  5.30E+5nMAssay Description:Inhibition of MAO-B in bovine brain mitochondria using benzylamine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088566(CHEMBL3577039)
Affinity DataIC50:  5.90E+5nMAssay Description:Inhibition of MAO-B in bovine brain mitochondria using benzylamine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088559(CHEMBL3577046)
Affinity DataIC50:  5.90E+5nMAssay Description:Inhibition of MAO-B in bovine brain mitochondria using benzylamine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088565(CHEMBL3577040)
Affinity DataIC50:  7.30E+5nMAssay Description:Inhibition of MAO-B in bovine brain mitochondria using benzylamine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088558(CHEMBL3577047)
Affinity DataIC50:  7.80E+5nMAssay Description:Inhibition of MAO-B in bovine brain mitochondria using benzylamine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088561(CHEMBL3577044)
Affinity DataIC50:  7.90E+5nMAssay Description:Inhibition of MAO-B in bovine brain mitochondria using benzylamine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088558(CHEMBL3577047)
Affinity DataIC50:  9.30E+5nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088567(CHEMBL3577038)
Affinity DataIC50:  9.50E+5nMAssay Description:Inhibition of MAO-B in bovine brain mitochondria using benzylamine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088556(CHEMBL3577034)
Affinity DataIC50:  9.90E+5nMAssay Description:Inhibition of MAO-B in bovine brain mitochondria using benzylamine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088568(CHEMBL3577037)
Affinity DataIC50:  9.90E+5nMAssay Description:Inhibition of MAO-B in bovine brain mitochondria using benzylamine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed