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Found 33 Enz. Inhib. hit(s) with all data for entry = 50044982
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040212(CHEMBL3359473)
Affinity DataIC50:  400nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040200(CHEMBL3359485)
Affinity DataIC50:  750nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040204(CHEMBL3359481)
Affinity DataIC50:  750nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040107(CHEMBL3359496)
Affinity DataIC50:  890nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040213(CHEMBL3359472)
Affinity DataIC50:  900nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040207(CHEMBL3359478)
Affinity DataIC50:  990nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040160(CHEMBL3359492)
Affinity DataIC50:  1.03E+3nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040164(CHEMBL3359489)
Affinity DataIC50:  1.05E+3nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040211(CHEMBL3359474)
Affinity DataIC50:  1.12E+3nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040214(CHEMBL3359471)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040118(CHEMBL3359495)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040205(CHEMBL3359480)
Affinity DataIC50:  1.49E+3nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040122(CHEMBL3359494)
Affinity DataIC50:  1.52E+3nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040201(CHEMBL3359484)
Affinity DataIC50:  1.56E+3nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040209(CHEMBL3359476)
Affinity DataIC50:  1.61E+3nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040206(CHEMBL3359479)
Affinity DataIC50:  1.61E+3nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040163(CHEMBL3359490)
Affinity DataIC50:  1.66E+3nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  2.08E+3nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040208(CHEMBL3359477)
Affinity DataIC50:  2.38E+3nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040215(CHEMBL3359470)
Affinity DataIC50:  2.52E+3nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040210(CHEMBL3359475)
Affinity DataIC50:  2.87E+3nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040172(CHEMBL3359488)
Affinity DataIC50:  3.31E+3nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040180(CHEMBL3359487)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040157(CHEMBL3359493)
Affinity DataIC50:  4.63E+3nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040162(CHEMBL3359491)
Affinity DataIC50:  4.74E+3nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040203(CHEMBL3359482)
Affinity DataIC50:  4.81E+3nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040186(CHEMBL3359486)
Affinity DataIC50:  5.93E+3nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040218(CHEMBL3359467)
Affinity DataIC50:  1.11E+4nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040219(CHEMBL3359466)
Affinity DataIC50:  1.35E+4nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040202(CHEMBL3359483)
Affinity DataIC50:  1.37E+4nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040217(CHEMBL3359468)
Affinity DataIC50:  3.55E+4nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50040216(CHEMBL3359469)
Affinity DataIC50:  1.86E+5nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50580((2Z)-2-(3,4-dihydroxybenzylidene)-6-hydroxy-coumar...)
Affinity DataIC50:  6.99E+5nMAssay Description:Inhibition of ICR mouse brain AChE using acetylthiocholine iodide as substrate preincubated for 10 mins before substrate addition by modified Ellman'...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed