Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 5697
TargetBeta-adrenergic receptor kinase 1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

LigandPNGBDBM84342(4-[1-hydroxy-2-(methylamino)ethyl]benzene-1,2-diol...)
Affinity DataKd:  610nMAssay Description:The binding of ligands to wild-type beta-AR was measured by competition with 35 pM 125I-CYP.More data for this Ligand-Target Pair
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TargetBeta-adrenergic receptor kinase 1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

LigandPNGBDBM25392(4-[1-hydroxy-2-(isopropylamino)ethyl]pyrocatechol;...)
Affinity DataKd:  200nMAssay Description:The binding of ligands to wild-type beta-AR was measured by competition with 35 pM 125I-CYP.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-adrenergic receptor kinase 1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

LigandPNGBDBM46041(1-(3,4-dihydroxyphenyl)-2-(isopropylamino)ethanone...)
Affinity DataKd:  9.00E+5nMAssay Description:The binding of ligands to wild-type beta-AR was measured by competition with 35 pM 125I-CYP.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-adrenergic receptor kinase 1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

LigandPNGBDBM92680(4-{1-hydroxy-2-[(propan-2-yl)amino]ethyl}phenol, 8)
Affinity DataKd:  5.20E+3nMAssay Description:The binding of ligands to wild-type beta-AR was measured by competition with 35 pM 125I-CYP.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-adrenergic receptor kinase 1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

LigandPNGBDBM25770(5-[2-(tert-butylamino)-1-hydroxyethyl]benzene-1,3-...)
Affinity DataKd:  7.40E+3nMAssay Description:The binding of ligands to wild-type beta-AR was measured by competition with 35 pM 125I-CYP.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-adrenergic receptor kinase 1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

LigandPNGBDBM50295572(5-(1-Hydroxy-2-isopropylamino-ethyl)-benzene-1,3-d...)
Affinity DataKd:  1.30E+4nMAssay Description:The binding of ligands to wild-type beta-AR was measured by competition with 35 pM 125I-CYP.More data for this Ligand-Target Pair
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TargetBeta-adrenergic receptor kinase 1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

LigandPNGBDBM92679(3-{1-hydroxy-2-[(propan-2-yl)amino]ethyl}phenol, 7)
Affinity DataKd:  3.00E+4nMAssay Description:The binding of ligands to wild-type beta-AR was measured by competition with 35 pM 125I-CYP.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-adrenergic receptor kinase 1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

LigandPNGBDBM92678(2-(tert-butylamino)-1-phenylethan-1-ol, 4)
Affinity DataKd:  4.10E+3nMAssay Description:The binding of ligands to wild-type beta-AR was measured by competition with 35 pM 125I-CYP.More data for this Ligand-Target Pair
In DepthDetails PubMed