Compile Data Set for Download or QSAR
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Found 8 Enz. Inhib. hit(s) with all data for entry = 50045012
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50041550(CHEMBL3358413)
Affinity DataIC50:  3.30nMAssay Description:Antagonist activity against human GnRH receptor expressed in CHO cells by IP-one HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50041550(CHEMBL3358413)
Affinity DataIC50:  3.30nMAssay Description:Antagonist activity against human GnRH receptor expressed in CHO cells by IP-one HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50041552(CHEMBL3358415)
Affinity DataIC50:  68nMAssay Description:Antagonist activity against human GnRH receptor expressed in CHO cells by IP-one HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50041552(CHEMBL3358415)
Affinity DataIC50:  68nMAssay Description:Antagonist activity against human GnRH receptor expressed in CHO cells by IP-one HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50041551(CHEMBL3358414)
Affinity DataIC50:  107nMAssay Description:Antagonist activity against human GnRH receptor expressed in CHO cells by IP-one HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50041551(CHEMBL3358414)
Affinity DataIC50:  107nMAssay Description:Antagonist activity against human GnRH receptor expressed in CHO cells by IP-one HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50041553(CHEMBL3358416)
Affinity DataIC50:  9.35E+3nMAssay Description:Antagonist activity against human GnRH receptor expressed in CHO cells by IP-one HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50041553(CHEMBL3358416)
Affinity DataIC50:  9.35E+3nMAssay Description:Antagonist activity against human GnRH receptor expressed in CHO cells by IP-one HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed