Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with all data for entry = 50045835
TargetNuclear factor NF-kappa-B p105 subunit(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50084420(CHEMBL3263013)
Affinity DataIC50:  1.11E+4nMAssay Description:Inhibition of TNF-alpha-stimulated NF-kappaB p50 (unknown origin) expressed in HEK293 cells preincubated for 4 hrs followed by TNF-alpha challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear factor NF-kappa-B p105 subunit(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50084419(Andrographolide | CHEBI:65408)
Affinity DataIC50:  4.96E+4nMAssay Description:Inhibition of TNF-alpha-stimulated NF-kappaB p50 (unknown origin) expressed in HEK293 cells preincubated for 4 hrs followed by TNF-alpha challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed