Compile Data Set for Download or QSAR
maximum 50k data
Found 18 Enz. Inhib. hit(s) with all data for entry = 6749
TargetCathepsin B(Capra hircus (Goat))
Kurukshetra University

LigandPNGBDBM150783(2-(4-Fluorophenyl)-2,3-dihydroquinazolin-4(1H)-one...)
Affinity DataKi:  6.40nMpH: 6.0Assay Description:Cathepsin B and H were first activated in the presence of thiol activators at pH 6.0 and pH 7.0, respectively. Then, 15 無 of the enzyme solution was...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Capra hircus (Goat))
Kurukshetra University

LigandPNGBDBM150782(2-(4-Chlorophenyl)-2,3-dihydroquinazolin-4(1H)-one...)
Affinity DataKi:  41nMpH: 6.0Assay Description:Cathepsin B and H were first activated in the presence of thiol activators at pH 6.0 and pH 7.0, respectively. Then, 15 無 of the enzyme solution was...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Capra hircus (Goat))
Kurukshetra University

LigandPNGBDBM150779(2-(4-Nitrophenyl)-2,3-dihydroquinazolin-4(1H)-one ...)
Affinity DataKi:  1.57E+3nMpH: 6.0Assay Description:Cathepsin B and H were first activated in the presence of thiol activators at pH 6.0 and pH 7.0, respectively. Then, 15 無 of the enzyme solution was...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin H(Capra hircus (Goat))
Kurukshetra University

LigandPNGBDBM150780(2-(4-Methylphenyl)-2,3-dihydroquinazolin-4(1H)-one...)
Affinity DataKi:  2.50E+3nMpH: 6.0Assay Description:Cathepsin B and H were first activated in the presence of thiol activators at pH 6.0 and pH 7.0, respectively. Then, 15 無 of the enzyme solution was...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Capra hircus (Goat))
Kurukshetra University

LigandPNGBDBM150781(2-(4-Methoxyphenyl)-2,3-dihydroquinazolin-4(1H)-on...)
Affinity DataKi:  2.81E+3nMpH: 6.0Assay Description:Cathepsin B and H were first activated in the presence of thiol activators at pH 6.0 and pH 7.0, respectively. Then, 15 無 of the enzyme solution was...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin H(Capra hircus (Goat))
Kurukshetra University

LigandPNGBDBM150783(2-(4-Fluorophenyl)-2,3-dihydroquinazolin-4(1H)-one...)
Affinity DataKi:  8.18E+3nMpH: 6.0Assay Description:Cathepsin B and H were first activated in the presence of thiol activators at pH 6.0 and pH 7.0, respectively. Then, 15 無 of the enzyme solution was...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin H(Capra hircus (Goat))
Kurukshetra University

LigandPNGBDBM150779(2-(4-Nitrophenyl)-2,3-dihydroquinazolin-4(1H)-one ...)
Affinity DataKi:  1.04E+4nMpH: 6.0Assay Description:Cathepsin B and H were first activated in the presence of thiol activators at pH 6.0 and pH 7.0, respectively. Then, 15 無 of the enzyme solution was...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Capra hircus (Goat))
Kurukshetra University

LigandPNGBDBM150784(2-(4-(Dimethylamino)phenyl)-2,3-dihydroquinazolin-...)
Affinity DataKi:  1.06E+4nMpH: 6.0Assay Description:Cathepsin B and H were first activated in the presence of thiol activators at pH 6.0 and pH 7.0, respectively. Then, 15 無 of the enzyme solution was...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin H(Capra hircus (Goat))
Kurukshetra University

LigandPNGBDBM50106307(2-Phenyl-2,3-dihydro-1H-quinazolin-4-one | CHEMBL1...)
Affinity DataKi:  1.44E+4nMpH: 6.0Assay Description:Cathepsin B and H were first activated in the presence of thiol activators at pH 6.0 and pH 7.0, respectively. Then, 15 無 of the enzyme solution was...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Capra hircus (Goat))
Kurukshetra University

LigandPNGBDBM150785(1H-Spiro(cyclohexane-1,2-quinazolin)-4(3H)-one (1i...)
Affinity DataKi:  1.50E+4nMpH: 6.0Assay Description:Cathepsin B and H were first activated in the presence of thiol activators at pH 6.0 and pH 7.0, respectively. Then, 15 無 of the enzyme solution was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin H(Capra hircus (Goat))
Kurukshetra University

LigandPNGBDBM150784(2-(4-(Dimethylamino)phenyl)-2,3-dihydroquinazolin-...)
Affinity DataKi:  1.86E+4nMpH: 6.0Assay Description:Cathepsin B and H were first activated in the presence of thiol activators at pH 6.0 and pH 7.0, respectively. Then, 15 無 of the enzyme solution was...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin H(Capra hircus (Goat))
Kurukshetra University

LigandPNGBDBM150782(2-(4-Chlorophenyl)-2,3-dihydroquinazolin-4(1H)-one...)
Affinity DataKi:  2.33E+4nMpH: 6.0Assay Description:Cathepsin B and H were first activated in the presence of thiol activators at pH 6.0 and pH 7.0, respectively. Then, 15 無 of the enzyme solution was...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Capra hircus (Goat))
Kurukshetra University

LigandPNGBDBM100101(2-(4-Bromo-phenyl)-2,3-dihydro-1H-quinazolin-4-one...)
Affinity DataKi:  3.25E+4nMpH: 6.0Assay Description:Cathepsin B and H were first activated in the presence of thiol activators at pH 6.0 and pH 7.0, respectively. Then, 15 無 of the enzyme solution was...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Capra hircus (Goat))
Kurukshetra University

LigandPNGBDBM150780(2-(4-Methylphenyl)-2,3-dihydroquinazolin-4(1H)-one...)
Affinity DataKi:  5.26E+4nMpH: 6.0Assay Description:Cathepsin B and H were first activated in the presence of thiol activators at pH 6.0 and pH 7.0, respectively. Then, 15 無 of the enzyme solution was...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin H(Capra hircus (Goat))
Kurukshetra University

LigandPNGBDBM100101(2-(4-Bromo-phenyl)-2,3-dihydro-1H-quinazolin-4-one...)
Affinity DataKi:  5.26E+4nMpH: 6.0Assay Description:Cathepsin B and H were first activated in the presence of thiol activators at pH 6.0 and pH 7.0, respectively. Then, 15 無 of the enzyme solution was...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin H(Capra hircus (Goat))
Kurukshetra University

LigandPNGBDBM150781(2-(4-Methoxyphenyl)-2,3-dihydroquinazolin-4(1H)-on...)
Affinity DataKi:  5.68E+4nMpH: 6.0Assay Description:Cathepsin B and H were first activated in the presence of thiol activators at pH 6.0 and pH 7.0, respectively. Then, 15 無 of the enzyme solution was...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin H(Capra hircus (Goat))
Kurukshetra University

LigandPNGBDBM150785(1H-Spiro(cyclohexane-1,2-quinazolin)-4(3H)-one (1i...)
Affinity DataKi:  9.01E+4nMpH: 6.0Assay Description:Cathepsin B and H were first activated in the presence of thiol activators at pH 6.0 and pH 7.0, respectively. Then, 15 無 of the enzyme solution was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin B(Capra hircus (Goat))
Kurukshetra University

LigandPNGBDBM50106307(2-Phenyl-2,3-dihydro-1H-quinazolin-4-one | CHEMBL1...)
Affinity DataKi:  1.11E+5nMpH: 6.0Assay Description:Cathepsin B and H were first activated in the presence of thiol activators at pH 6.0 and pH 7.0, respectively. Then, 15 無 of the enzyme solution was...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed