Affinity DataIC50: 10nMAssay Description:Inhibition of BRD4 bromodomain 1 (unknown origin) incubated in dark for 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Glaxosmithkline R&D
Curated by ChEMBL
Glaxosmithkline R&D
Curated by ChEMBL
Affinity DataIC50: 196nMAssay Description:Inhibition of BRD3 in human HUT78 cells incubated for 45 mins by chemoproteomic competition binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.05E+3nMAssay Description:Binding affinity to partial length human BRD7 by BROMOscan assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of BRD9 in human HUT78 cells incubated for 45 mins by chemoproteomic competition binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibition of BRD4 bromodomain 1 (unknown origin) incubated in dark for 30 mins by TR-FRET assayMore data for this Ligand-Target Pair