Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50046098
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Acelot

Curated by ChEMBL
LigandPNGBDBM50094871(CHEMBL3590142)
Affinity DataIC50:  450nMAssay Description:Inhibition of LRRK2 G2019S mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Acelot

Curated by ChEMBL
LigandPNGBDBM50094873(CHEMBL3588873)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of LRRK2 G2019S mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Acelot

Curated by ChEMBL
LigandPNGBDBM50094872(CHEMBL3590143)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of LRRK2 G2019S mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Acelot

Curated by ChEMBL
LigandPNGBDBM50094872(CHEMBL3590143)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of wild type LRRK2 (unknown origin) assessed as inhibition of LRRKtide phosphorylation after 120 mins by radiometric assay in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Acelot

Curated by ChEMBL
LigandPNGBDBM50434582(CHEMBL2386594)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of LRRK2 G2019S mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Acelot

Curated by ChEMBL
LigandPNGBDBM50434582(CHEMBL2386594)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of wild type LRRK2 (unknown origin) assessed as inhibition of LRRKtide phosphorylation after 120 mins by radiometric assay in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Acelot

Curated by ChEMBL
LigandPNGBDBM50094873(CHEMBL3588873)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of wild type LRRK2 (unknown origin) assessed as inhibition of LRRKtide phosphorylation after 120 mins by radiometric assay in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Acelot

Curated by ChEMBL
LigandPNGBDBM50094871(CHEMBL3590142)
Affinity DataIC50:  1.11E+4nMAssay Description:Inhibition of wild type LRRK2 (unknown origin) assessed as inhibition of LRRKtide phosphorylation after 120 mins by radiometric assay in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed