Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50046516
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50116793(CHEMBL3612750)
Affinity DataIC50:  2.16E+4nMAssay Description:Inhibition of His6-tagged Src kinase domain (unknown origin) using AEEEIYGEFEAKKKK as substrate preincubated for 10 mins followed by substrate/ATP ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM83209(7-amino-4-(trifluoromethyl)-1-benzopyran-2-one | 7...)
Affinity DataIC50:  3.09E+4nMAssay Description:Inhibition of His6-tagged Src kinase domain (unknown origin) using AEEEIYGEFEAKKKK as substrate preincubated for 10 mins followed by substrate/ATP ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50116794(CHEMBL3612749)
Affinity DataIC50:  3.65E+4nMAssay Description:Inhibition of His6-tagged Src kinase domain (unknown origin) using AEEEIYGEFEAKKKK as substrate preincubated for 10 mins followed by substrate/ATP ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50116792(CHEMBL3612751)
Affinity DataIC50:  7.35E+4nMAssay Description:Inhibition of His6-tagged Src kinase domain (unknown origin) using AEEEIYGEFEAKKKK as substrate preincubated for 10 mins followed by substrate/ATP ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed