Compile Data Set for Download or QSAR
maximum 50k data
Found 25 Enz. Inhib. hit(s) with all data for entry = 50046608
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121214(CHEMBL3623075)
Affinity DataKi:  140nMAssay Description:Displacement of [125I]orexin-A from human OX1R expressed in CHO cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121214(CHEMBL3623075)
Affinity DataKi:  770nMAssay Description:Displacement of [125I]orexin-A from human OX2R expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121217(CHEMBL3622420)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human OX2R expressed in CHOK1 cells by NFAT-response luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121218(CHEMBL3622421)
Affinity DataEC50:  182nMAssay Description:Agonist activity at human OX2R expressed in CHOK1 cells by NFAT-response luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121219(CHEMBL3622422)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human OX2R expressed in CHOK1 cells by NFAT-response luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121220(CHEMBL3622423)
Affinity DataEC50:  235nMAssay Description:Agonist activity at human OX2R expressed in CHOK1 cells by NFAT-response luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121221(CHEMBL3622424)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human OX2R expressed in CHOK1 cells by NFAT-response luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121262(CHEMBL3622425)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human OX2R expressed in CHOK1 cells by NFAT-response luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121265(CHEMBL3622426)
Affinity DataEC50:  268nMAssay Description:Agonist activity at human OX2R expressed in CHOK1 cells by NFAT-response luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121306(CHEMBL3622427)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human OX2R expressed in CHOK1 cells by NFAT-response luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121323(CHEMBL3623079)
Affinity DataEC50:  2.75E+3nMAssay Description:Agonist activity at human OX1R expressed in CHOK1 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121308(CHEMBL3622429)
Affinity DataEC50:  1.05E+3nMAssay Description:Agonist activity at human OX2R expressed in CHOK1 cells by NFAT-response luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121309(CHEMBL3623074)
Affinity DataEC50:  800nMAssay Description:Agonist activity at human OX2R expressed in CHOK1 cells by NFAT-response luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121214(CHEMBL3623075)
Affinity DataEC50:  23nMAssay Description:Agonist activity at human OX2R expressed in CHOK1 cells by NFAT-response luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121310(CHEMBL3623076)
Affinity DataEC50:  31nMAssay Description:Agonist activity at human OX2R expressed in CHOK1 cells by NFAT-response luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121311(CHEMBL3623077)
Affinity DataEC50:  94nMAssay Description:Agonist activity at human OX2R expressed in CHOK1 cells by NFAT-response luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121323(CHEMBL3623079)
Affinity DataEC50:  28nMAssay Description:Agonist activity at human OX2R expressed in CHOK1 cells by NFAT-response luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121219(CHEMBL3622422)
Affinity DataEC50:  5.23E+3nMAssay Description:Agonist activity at human OX1R expressed in CHOK1 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121307(CHEMBL3622428)
Affinity DataEC50:  9.25E+3nMAssay Description:Agonist activity at human OX1R expressed in CHOK1 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121214(CHEMBL3623075)
Affinity DataEC50:  1.62E+3nMAssay Description:Agonist activity at human OX1R expressed in CHOK1 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121310(CHEMBL3623076)
Affinity DataEC50:  6.13E+3nMAssay Description:Agonist activity at human OX1R expressed in CHOK1 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121311(CHEMBL3623077)
Affinity DataEC50:  5.72E+3nMAssay Description:Agonist activity at human OX1R expressed in CHOK1 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121216(CHEMBL3622419)
Affinity DataEC50:  800nMAssay Description:Agonist activity at human OX2R expressed in CHOK1 cells by NFAT-response luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121215(CHEMBL3621218)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human OX2R expressed in CHOK1 cells by NFAT-response luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121307(CHEMBL3622428)
Affinity DataEC50:  33nMAssay Description:Agonist activity at human OX2R expressed in CHOK1 cells by NFAT-response luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed