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Found 9 Enz. Inhib. hit(s) with all data for entry = 50046719
TargetMu-type opioid receptor(Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50127701(CHEMBL3627737)
Affinity DataKi:  0.515nMAssay Description:Displacement of [3H]-DAMGO from mu opioid receptor (unknown origin) transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50127700(CHEMBL3629337)
Affinity DataKi:  0.565nMAssay Description:Displacement of [3H]-DAMGO from mu opioid receptor (unknown origin) transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50095155((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]-DAMGO from mu opioid receptor (unknown origin) transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50095155((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataKi:  6.08E+3nMAssay Description:Displacement of [3H]-DPDPE from delta opioid receptor (unknown origin) transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50127700(CHEMBL3629337)
Affinity DataKi:  1.21E+4nMAssay Description:Displacement of [3H]-DPDPE from delta opioid receptor (unknown origin) transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50127701(CHEMBL3627737)
Affinity DataKi:  1.33E+4nMAssay Description:Displacement of [3H]-DPDPE from delta opioid receptor (unknown origin) transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50095155((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataEC50:  14nMAssay Description:Agonist activity at mu opioid receptor (unknown origin) transfected in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50127700(CHEMBL3629337)
Affinity DataEC50:  0.0629nMAssay Description:Agonist activity at mu opioid receptor (unknown origin) transfected in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50127701(CHEMBL3627737)
Affinity DataEC50:  0.0643nMAssay Description:Agonist activity at mu opioid receptor (unknown origin) transfected in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed