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Found 42 Enz. Inhib. hit(s) with all data for entry = 50046789
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)
Affinity DataIC50:  7.60nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataIC50:  13nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131218(CHEMBL3634406)
Affinity DataIC50:  14nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131175(CHEMBL3634540)
Affinity DataIC50:  18nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131176(CHEMBL3634539)
Affinity DataIC50:  31nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131215(CHEMBL3634409)
Affinity DataIC50:  84nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131217(CHEMBL3634407)
Affinity DataIC50:  86nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131214(CHEMBL3634530)
Affinity DataIC50:  180nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)
Affinity DataIC50:  220nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131172(CHEMBL3634543)
Affinity DataIC50:  250nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataIC50:  340nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131218(CHEMBL3634406)
Affinity DataIC50:  450nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131174(CHEMBL3634541)
Affinity DataIC50:  450nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131214(CHEMBL3634530)
Affinity DataIC50:  740nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131176(CHEMBL3634539)
Affinity DataIC50:  1.04E+3nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131184(CHEMBL3634535)
Affinity DataIC50:  1.89E+3nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131217(CHEMBL3634407)
Affinity DataIC50:  2.07E+3nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131191(CHEMBL3634534)
Affinity DataIC50:  2.37E+3nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131212(CHEMBL3634531)
Affinity DataIC50:  2.76E+3nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131215(CHEMBL3634409)
Affinity DataIC50:  3.41E+3nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131178(CHEMBL3634537)
Affinity DataIC50:  8.56E+3nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131177(CHEMBL3634538)
Affinity DataIC50:  1.43E+4nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131179(CHEMBL3634536)
Affinity DataIC50:  2.28E+4nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131175(CHEMBL3634540)
Affinity DataIC50:  2.88E+4nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131216(CHEMBL3634408)
Affinity DataIC50:  4.92E+4nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131174(CHEMBL3634541)
Affinity DataIC50:  5.63E+4nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131184(CHEMBL3634535)
Affinity DataIC50:  6.56E+4nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131177(CHEMBL3634538)
Affinity DataIC50:  7.53E+4nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131211(CHEMBL3634532)
Affinity DataIC50:  8.35E+4nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131212(CHEMBL3634531)
Affinity DataIC50:  9.46E+4nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131213(CHEMBL3632643)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Bcr-Abl T315I mutant (unknown origin) by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131211(CHEMBL3634532)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131173(CHEMBL3634542)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131172(CHEMBL3634543)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131065(CHEMBL3634544)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131065(CHEMBL3634544)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131216(CHEMBL3634408)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131179(CHEMBL3634536)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131178(CHEMBL3634537)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131210(CHEMBL3634533)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of wild type Bcr-Abl (unknown origin) by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131191(CHEMBL3634534)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
First Affiliated Hospital Of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50131210(CHEMBL3634533)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against interleukin-2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed